Title of article
PhI(OAc)2 and BF3–OEt2 mediated heterocyclization: metal-free synthesis of pyrimidine-annulated oxazolines
Author/Authors
Mondal، نويسنده , , Biplab and Hazra، نويسنده , , Somjit and Naktode، نويسنده , , Kishor and Panda، نويسنده , , Tarun K. and Roy، نويسنده , , B.، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2014
Pages
4
From page
5625
To page
5628
Abstract
A simple high yielding and highly efficient synthesis of oxazoline ring fused with uracil moiety is reported. Hypervalent iodine (PIDA) in the presence of BF3–OEt2 generates an effective electrophile to activate uracil C5–C6 double bond leading to heterocyclization.
Keywords
oxazoline , hypervalent iodine , Pyrimidine , BF3–OEt2 , cyclization , PhI(OAc)2
Journal title
Tetrahedron Letters
Serial Year
2014
Journal title
Tetrahedron Letters
Record number
1890851
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