Title of article :
Expedient BINOL derivative arylations
Author/Authors :
Albini، نويسنده , , Mathieu and Taillier، نويسنده , , Catherine and Dalla، نويسنده , , Vincent and Blanchet، نويسنده , , Jérôme and Rouden، نويسنده , , Jacques، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2014
Abstract :
A dramatic improvement of our previous methodology based on a Suzuki–Miyaura cross-coupling to access 3,3′-disubstituted H8-BINOLs using microwave heating is reported herein. These new conditions represent a large gain in term of atom-economy, reaction time, catalyst loading, and excess of reagents employed.
Keywords :
PALLADIUM , Suzuki coupling , microwave , Binol , arylation
Journal title :
Tetrahedron Letters
Journal title :
Tetrahedron Letters