• Title of article

    High-Yielding Synthesis of 3-Alkoxycarbonyl- and 3-Carboxamido-3-tropene Derivatives in Homogeneous Carbonylation Reactions of 3-Iodo-2-tropene

  • Author/Authors

    Horváth, László University of Pécs - Department of Inorganic Chemistry, Hungary , Horváth, László MTA-PTE Research Group for Chemical Sensors, Hungary , Berente, Zoltán University of Pécs - Department of Inorganic Chemistry, Hungary , Berente, Zoltán MTA-PTE Research Group for Chemical Sensors, Hungary , Kollár, László University of Pécs - Department of Inorganic Chemistry, Hungary , Kollár, László MTA-PTE Research Group for Chemical Sensors, Hungary

  • From page
    124
  • To page
    127
  • Abstract
    3-Iodo-2-tropene, synthesized from the corresponding ketone (tropinone) via its hydrazone, wascarbonylated in palladium-catalyzed alkoxy- and aminocarbonylation reactions. The new synthetic approach provided the corresponding 3-carboxylic acid derivatives of pharmacological importance in chemospecific reactions and isolated in up to 87 % yields.
  • Keywords
    Tropane , skeleton , palladium , aminocarbonylation , alkoxycarbonylation , homogeneous catalysis
  • Journal title
    letters in organic chemistry
  • Journal title
    letters in organic chemistry
  • Record number

    2717824