• Title of article

    FPL 64176: The effect of the chain length separating the two aryl groups on calcium agonist activity

  • Author/Authors

    John M. Kane، نويسنده , , Christopher R. Dalton، نويسنده , , Nelson L. Velayo، نويسنده , , David Rampe، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1995
  • Pages
    4
  • From page
    873
  • To page
    876
  • Abstract
    Analogs of the L-type calcium channel agonist FPL 64176 (5) were prepared in which the chain length separating the two aryl moieties was varied between zero and four. FPL 64176 (5) and phenethyl derivative 19 were the most potent compounds tested, displaying EC50 values for enhancing calcium influx into GH3 cells of 1−2×10−7 M.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1995
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    787434