• Title of article

    A novel non nucleoside compound with high in vitro anti-HIV-1 activity. Absolute stereochemistry determination

  • Author/Authors

    De la Fuente Jes?s A.، نويسنده , , Marug?n Juan J.، نويسنده , , Cross Sue S.، نويسنده , , Mateos Alfonso F.، نويسنده , , A. Garcia Santiago، نويسنده , , Menéndez Amador، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1995
  • Pages
    4
  • From page
    1471
  • To page
    1474
  • Abstract
    Here we report a novel non-nucleoside compound, PM-92131(+), with in vitro anti-HIV-1 activity. This product was synthesized as a pure enantiomer via diastereomeric ester formation and selective crystallisation and its absolute stereochemistry was determined by X-ray diffraction analysis. Results from the activity assays suggest PM-92131(+) could be a promising new compound for further assessment as a potential anti-HIV-1 agent.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1995
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    787543