Title of article
4-bromo-1-methoxy-N-[2-(4-aryl-1-piperazinyl)ethyl]-2-naphthalenecarboxamides: Selective dopamine D3 receptor partial agonists
Author/Authors
Shelly A. Glase، نويسنده , , Hyacinth C. Akunne، نويسنده , , Thomas G. Heffner، نويسنده , , Stephen J. Johnson، نويسنده , , Suzanne R. Kesten، نويسنده , , Robert G. MacKenzie، نويسنده , , Peter J. Manley، نويسنده , , Thomas A. Pugsley، نويسنده , , Jon L. Wright، نويسنده , , Lawrence D. Wise، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 1996
Pages
6
From page
1361
To page
1366
Abstract
A series of 4-bromo-1-methoxy-N-[2-(4-aryl-1-piperazinyl)ethyl]-2-naphthalenecarboxamide dopamine (DA) D3 receptor agonists has been identified. These compounds were found to be selective for DA D3 over D2 receptors and were shown to be partial to full agonists as measured by stimulation of mitogenesis in D3-transfected CHO p-5 cells.
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
1996
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
788119
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