Title of article
BMS-187257, a potent, selective, and novel heterocyclic β3 adrenergic receptor agonist
Author/Authors
Liesl G. Fisher، نويسنده , , Philip M. Sher، نويسنده , , Stephen Skwish، نويسنده , , Inge M. Michel، نويسنده , , Steven M. Seiler، نويسنده , , Kenneth E. J. Dickinson، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 1996
Pages
6
From page
2253
To page
2258
Abstract
Novel heterocyclic β3 adrenergic receptor agonists2 were prepared and evaluated for their ability to bind to human β1, β2, and β3 adrenergic receptors. Stimulatory effects on the β3 adrenergic receptor were also measured. BMS-187257 (4b) was found to be a potent and selective β3 agonist.
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
1996
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
788334
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