• Title of article

    Synthesis and antibacterial activity of lipophilic carbapenems with anti-MRSA activity

  • Author/Authors

    Jean Claude Arnould، نويسنده , , Ruth N Illingworth، نويسنده , , Wright W Nichols، نويسنده , , R. Geoffrey Wilson، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1996
  • Pages
    6
  • From page
    2449
  • To page
    2454
  • Abstract
    A series of sulphur-linked and carbon-linked lipophilic carbapenems has been prepared and evaluated for antibacterial activity in vitro and in vivo and for affinity for PBP2′ of Staphylococcus aureus. Potent activity in vitro against methicillin-resistant S. aureus and methicillin-resistant coagulase negative staphylococci was observed despite IC50 values for PBP2′ being higher than the MIC.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1996
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    788374