• Title of article

    Synthesis of novel ellipticine analogues and their inhibition of Moloney leukaemia reverse transcriptase

  • Author/Authors

    Géza Tim?ri، نويسنده , , Tibor So?s، نويسنده , , Gyorgy Hajos، نويسنده , , Andr?s Messmer، نويسنده , , J?nos Nacsa، نويسنده , , Jozsef Molnar، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1996
  • Pages
    6
  • From page
    2831
  • To page
    2836
  • Abstract
    Two new ellipticine analogues were synthetized as potential non nucleoside inhibitors of reverse transcriptase and were tested on Moloney leukaemia virus reverse transcriptase in vitro. Both derivatives (9a,b) showed considerable inhibitory effect; ID50 was found to be in the range of 2.8 to 4.5 × 10−5 M.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1996
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    788449