• Title of article

    Potent novel nonsteroidal androgen antagonists with a phthalimide skeleton

  • Author/Authors

    Hiroyuki Miyachi، نويسنده , , Akihiko Azuma، نويسنده , , Takuya Kitamoto، نويسنده , , Kozue Hayashi، نويسنده , , Shigeaki Kato، نويسنده , , Masafumi Koga، نويسنده , , Bunzo Sato، نويسنده , , Yuichi Hashimoto، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1997
  • Pages
    6
  • From page
    1483
  • To page
    1488
  • Abstract
    Anti-androgenic activity of various phthalimide analogs was evaluated based on inhibition of androgen-induced activation of nuclear androgen receptor (CAT assay) and on growth inhibition of the androgen-dependent clonal cell line SC-3. Some compounds showed very potent androgen-antagonistic activity.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1997
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    788794