Title of article
Selective inhibition of the chymotrypsin-like activity of the 20S proteasome by 5-methoxy-1-indanone dipeptide benzamides
Author/Authors
Robert T. Lum، نويسنده , , Marek G. Nelson، نويسنده , , Alison Joly، نويسنده , , Amy G. Horsma، نويسنده , , Gavin Lee، نويسنده , , Stephanie M. Meyer، نويسنده , , Michael M. Wick، نويسنده , , Steven R. Schow، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 1998
Pages
6
From page
209
To page
214
Abstract
Potent inhibitors of the 20S proteasome that contain a novel indanone head group coupled to di and tripeptides are described. These compounds are the first proteasome inhibitors have demonstrated high selectivity for the chymotrypsin-like activity of the 20S proteasome.
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
1998
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
789212
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