• Title of article

    Anti-malarial activities of acylated bruceolide derivatives

  • Author/Authors

    Nobutoshi Murakami، نويسنده , , Takashi Umezome، نويسنده , , Taifo Mahmud، نويسنده , , Masanori Sugimoto، نويسنده , , Motomasa Kobayashi، نويسنده , , Yusuke Wataya، نويسنده , , Hye Sook Kim، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1998
  • Pages
    4
  • From page
    459
  • To page
    462
  • Abstract
    Several O-acylated derivatives of bruceolide (2) were synthesized and their anti-malarial activities together with selective toxicities were examined. It was found that 3,15-di-O-acetyl- (3c), 3,15-di-O-propionyl- (3d) and 15-O-propionylbruceolide (3b), as well as bruceine B (3a), exhibited potent anti-malarial activities with high selective toxicities.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1998
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    789261