• Title of article

    Isoxazoline GPIIb/IIIa antagonists bearing a phosphoramidate

  • Author/Authors

    John Wityak، نويسنده , , A. Ewa Tobin، نويسنده , , Shaker A. Mousa، نويسنده , , Ruth R. Wexler، نويسنده , , Richard E. Olson، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1999
  • Pages
    4
  • From page
    123
  • To page
    126
  • Abstract
    Isoxazolinylacetamides bearing a phosphoramidate group α- to the carboxylate moiety (3) were prepared and evaluated for in vitro antiplatelet efficacy. They were found to bind GPIIb/IIIa with high affinity and were potent antagonists of ADP mediated platelet aggregation.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1999
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    789905