• Title of article

    Synthesis of tetrasubstituted bicyclo[3.2.1]octenes as potential inhibitors of influenza virus sialidase

  • Author/Authors

    Paul S. Jones، نويسنده , , Paul W. Smith، نويسنده , , George W. Hardy، نويسنده , , Peter D. Howes، نويسنده , , Richard J. Upton، نويسنده , , Richard C. Bethell، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1999
  • Pages
    6
  • From page
    605
  • To page
    610
  • Abstract
    Several racemic bicyclo[3.2.1]octene derivatives have been synthesised and evaluated as inhibitors of influenza virus sialidases. The 5-acetamido-bicyclo[3.2.1]octenol 4 showed modest activity against influenza A and B virus sialidases.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1999
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    790002