• Title of article

    Antimalarial activity of 3-hydroxyalkyl-2-methylene-propionic acid derivatives

  • Author/Authors

    Mrinal K. Kundu، نويسنده , , N. Sundar، نويسنده , , Srinivas K. Kumar، نويسنده , , Sujata V. Bhat، نويسنده , , Sukla Biswas، نويسنده , , Neena Valecha، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1999
  • Pages
    6
  • From page
    731
  • To page
    736
  • Abstract
    Several Baylis-Hillman adducts and their derivatives were synthesized and evaluated as targeted potential anti-malarials. The compounds 4, 7 and 9 were found to have highest potency against P. falciparum in vitro. The in vivo test result of compound 4 and 9 against P. berghei demonstrated activity at 80 mg/Kg dose level.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1999
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    790027