• Title of article

    The synthesis and in vitro cytotoxic studies of novel oxa-spermidine derivatives and homologues

  • Author/Authors

    Vladimir A. Kuksa، نويسنده , , Valentin A. Pavlov، نويسنده , , Paul Kong Thoo Lin، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2000
  • Pages
    3
  • From page
    1265
  • To page
    1267
  • Abstract
    A series of oxa-spermidine derivatives and homologues were prepared and their anticancer properties were evaluated. All these compounds showed an average GI50 value in the range of 3.9–28.9 μM. SAR studies showed that the presence of a sulphonamido functionality and the length of the alkyl chain are important factors for an enhanced activity.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2000
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    790848