• Title of article

    Bile acid–oligodeoxynucleotide conjugates: synthesis and liver excretion in rats

  • Author/Authors

    Dieter Starke، نويسنده , , Kerstin Lischka، نويسنده , , Peter Pagels، نويسنده , , Eugen Uhlmann، نويسنده , , Werner Kramer، نويسنده , , Günter Wess، نويسنده , , Ernst Petzinger، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2001
  • Pages
    5
  • From page
    945
  • To page
    949
  • Abstract
    The synthesis of bile acid–oligodeoxynucleotide conjugates via the 3-OH group of the bile acids is described. When used in vivo in rats, covalent conjugation of an oligodeoxynucleotide via a linker to cholic acid resulted in an increased biliary excretion of bile acid–oligodeoxynucleotide conjugates compared to unconjugated oligodeoxynucleotides.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2001
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    791312