• Title of article

    Increase of the adenallene anti-HIV activity in cell culture using its bis(tBuSATE) phosphotriester derivative

  • Author/Authors

    David Egron، نويسنده , , Christian Perigaud، نويسنده , , Gilles Gosselin، نويسنده , , Anne-Marie Aubertin، نويسنده , , Hiroyuki Gatanaga، نويسنده , , Hiroaki Mitsuya، نويسنده , , Jiri Zemlicka، نويسنده , , Jean-Louis Imbach، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2002
  • Pages
    2
  • From page
    265
  • To page
    266
  • Abstract
    The bis(S-pivaloyl-2-thioethyl) phosphotriester derivative of 9-(4′-hydroxy-1′,2′-butadienyl)adenine (adenallene) was synthesized. This mononucleotide prodrug proved to be more effective than the parent nucleoside in inhibiting HIV-1 replication in several human T4 lymphoblastoid cell lines.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2002
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    791949