• Title of article

    Alkylation of manganese(II) tetraphenylporphyrin by antimalarial fluorinated artemisinin derivatives

  • Author/Authors

    Montserrat Rodriguez، نويسنده , , Daniele Bonnet-Delpon، نويسنده , , Jean-Pierre Bégué، نويسنده , , Anne Robert، نويسنده , , Bernard Meunier، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2003
  • Pages
    4
  • From page
    1059
  • To page
    1062
  • Abstract
    The alkylating properties of two artemisinin derivatives bearing a trifluoromethyl substituent at C10 were evaluated toward manganese(II) tetraphenylporphyrin, considered as a heme model. Chlorin-type covalent adducts were obtained by alkylation of the porphyrin ring by C-centered radicals derived from reductive activation of the peroxide function of the drugs.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2003
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    793074