• Title of article

    Macrocyclic inhibitors of the bacterial cell wall biosynthesis enzyme mur D

  • Author/Authors

    James R. Horton، نويسنده , , Julieanne M. Bostock، نويسنده , , Ian Chopra، نويسنده , , Lars Hesse، نويسنده , , Simon E. V. Phillips، نويسنده , , David J. Adams and ...[et al.]، نويسنده , , A. Peter Johnson، نويسنده , , Colin W. G. Fishwick، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2003
  • Pages
    4
  • From page
    1557
  • To page
    1560
  • Abstract
    Computer-based molecular design has been used to produce a series of new macrocyclic systems targeted against the bacterial cell wall biosynthetic enzyme MurD. Following their preparation, which involved a novel metathesis-based cyclisation as the key step, these systems were found to show good inhibition when assayed against the MurD enzyme.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2003
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    793184