• Title of article

    Biological activities of α-mangostin derivatives against acidic sphingomyelinase

  • Author/Authors

    Motoko Hamada، نويسنده , , Kazuhiko Iikubo، نويسنده , , Yuichi Ishikawa، نويسنده , , Aya Ikeda، نويسنده , , Kazuo Umezawa، نويسنده , , Shigeru Nishiyama، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2003
  • Pages
    3
  • From page
    3151
  • To page
    3153
  • Abstract
    Deprenyl and benzofenone-type congeners of α-mangostin 1 have been synthesized to understand their role for the inhibitory activity against sphingomyelinase (SMase). While removal of the prenyl group of the right side (11 and 12) caused loss of the selectivity between ASMase (acidic sphingomyelinase) and NSMase (neutral sphingomyelinase), the prenyl group of the left side appeared to increase the inhibitory activities (16 and 17).
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2003
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    793527