Title of article
Fused pyrimidine based inhibitors of phosphodiesterase 7 (PDE7): synthesis and initial structure–activity relationships
Author/Authors
James Kempson، نويسنده , , William J. Pitts، نويسنده , , Joseph Barbosa، نويسنده , , Junqing Guo، نويسنده , , Omonike Omotoso، نويسنده , , Andrew Watson، نويسنده , , Karen Stebbins، نويسنده , , Gary C. Starling، نويسنده , , John H. Dodd، نويسنده , , Joel C. Barrish، نويسنده , , Raymond Felix، نويسنده , , Urs Karl Fischer، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 2005
Pages
5
From page
1829
To page
1833
Abstract
A series of fused pyrimidine based inhibitors of PDE7 have been derived from an earlier screening lead 1. The synthesis, structure–activity relationships (SAR) and selectivity against several other PDE family members are described.
Keywords
Pyrimidine , PDE7
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
2005
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
795487
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