Author/Authors :
Yutaka Aoyagi، نويسنده , , Yukio Hitotsuyanagi، نويسنده , , Tomoyo Hasuda، نويسنده , , Haruhiko Fukaya، نويسنده , , Koichi Takeya، نويسنده , , Ritsuo Aiyama، نويسنده , , Takeshi Matsuzaki، نويسنده , , Shusuke Hashimoto، نويسنده ,
Abstract :
Several C-ring modified analogues of a potent antileukemic diterpene, triptolide (1), were synthesized and their structure–activity relationships were studied.
Keywords :
antitumor , Structure–activity relationships , Semisynthesis , C-ring , Triptolide analogues