• Title of article

    Synthesis of biotinylated photoaffinity probes based on arylsulfonamide γ-secretase inhibitors

  • Author/Authors

    Haruhiko Fuwa، نويسنده , , Kenichi Hiromoto، نويسنده , , Yasuko Takahashi، نويسنده , , Satoshi Yokoshima، نويسنده , , Toshiyuki Kan، نويسنده , , Tohru Fukuyama، نويسنده , , Takeshi Iwatsubo، نويسنده , , Taisuke Tomita، نويسنده , , Hideaki Natsugari، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2006
  • Pages
    6
  • From page
    4184
  • To page
    4189
  • Abstract
    Synthesis and biological evaluation of an arylsulfonamide class of γ-secretase inhibitors are described. Design, synthesis, and biological evaluation of multifunctional molecular probes harboring a benzophenone photophore as a cross-linking group and a biotin tag are also reported.
  • Keywords
    Photoaffinity probes , ?-Secretase inhibitors , structure–activity relationships , Arylsulfonamides
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2006
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    797158