ليست عنوان مقالات لاتين Synthesis and antitumor activity of camptothecin derivatives bearing five-membered heterocycle containing 10-substituents Synthesis and biological evaluation of novel 3′-difluorovinyl taxoids

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1

Synthesis and antitumor activity of camptothecin derivatives bearing five-membered heterocycle containing 10-substituents

2

Synthesis and antitumor activity of certain 2,3,6-trisubstituted quinazolin-4(3H)-one derivatives

3

Synthesis and antitumor activity of cyclodepsipeptide zygosporamide and its analogues

4

Synthesis and antitumor activity of des-AB analogue of steroidal saponin OSW-1

5

Synthesis and antitumor activity of DNA binding cationic porphyrin–platinum(II) complexes

6

Synthesis and antitumor activity of duocarmycin derivatives: A-ring pyrrole analogues of duocarmycin B2 Original Research Article

7

Synthesis and antitumor activity of duocarmycin derivatives: A-ring pyrrole compounds bearing β-(5′,6′,7′-trimethoxy-2′-indolyl)acryloyl group Original Research Article

8

Synthesis and antitumor activity of duocarmycin derivatives: modification at C-8 position of A-ring pyrrole compounds bearing the simplified DNA-binding groups Original Research Article

9

Synthesis and antitumor activity of duocarmycin derivatives: modification at the C-7 position of segment-A of A-ring pyrrole compounds Original Research Article

10

Synthesis and antitumor activity of goniofufurone analogues Original Research Article

11

Synthesis and antitumor activity of icogenin and its analogue

12

Synthesis and antitumor activity of indolylpyrimidines: Marine natural product meridianin D analogues Original Research Article

13

Synthesis and antitumor activity of leinamycin derivatives: Modifications of C-8 hydroxy and C-9 keto groups

14

Synthesis and antitumor activity of new d-galactose-containing derivatives of doxorubicin Original Research Article

15

Synthesis and antitumor activity of novel 10-substituted camptothecin analogues Original Research Article

16

Synthesis and antitumor activity of novel C-8 ester derivatives of leinamycin

17

Synthesis and anti-tumor activity of novel combretastatins: combretocyclopentenones and related analogues

18

Synthesis and antitumor activity of novel cyclopropapyrroloindole (CPI) derivatives bearing bis(methoxycarbonyl) groups

19

Synthesis and antitumor activity of novel cyclopropapyrroloindole(CPI) derivatives bearing methoxycarbonyl and trifluoromethyl groups

20

Synthesis and antitumor activity of novel distamycin derivatives

21

Synthesis and antitumor activity of novel duocarmycin derivatives

22

Synthesis and antitumor activity of novel paclitaxel–chlorambucil hybrids

23

Synthesis and antitumor activity of selected 7-alkylidene substituted cephems Original Research Article

24

Synthesis and antitumor activity of simplified ecteinascidin–saframycin analogs

25

SYNTHESIS AND ANTITUMOR ACTIVITY OF SOME 5H-PYRROLIZINE, PYRIMIDO [5,4-a] PYRROLIZINE PYMMIDO[4,5-b]PYRROLIZINE DERIVATIVES

26

SYNTHESIS AND ANTITUMOR ACTIVITY OF SOME 5H-PYRROLIZINE, PYRIMIDO [5,4-a] PYRROLIZINE PYMMIDO[4,5-b]PYRROLIZINE DERIVATIVES

27

Synthesis and antitumor activity of some indeno[1,2-b]quinoline-based bis carboxamides Original Research Article

28

Synthesis and antitumor activity of some new pyrazolo[3,4-d]pyrimidine and pyrazolo[3,4-b]pyridine derivatives

29

Synthesis and antitumor activity of s-tetrazine derivatives

30

Synthesis and antitumor activity of the 7-O-(2,6-dideoxy-2-fluoro-α-l-talopyranosyl)daunomycinone derivatives modified at C-3′ or C-4′

31

Synthesis and antitumor activity of the hexacyclic camptothecin derivatives

32

Synthesis and antitumor activity of two natural N-acetylglucosamine-bearing triterpenoid saponins: Lotoidoside D and E

33

Synthesis and antitumor activity of water-soluble duocarmycin B1 prodrugs

34

Synthesis and antitumor activity of water-soluble enediyne compounds related to dynemicin a Original Research Article

35

Synthesis and anti-tumor activity of β-C-glycoside analogs of the immunostimulant KRN7000

36

Synthesis and antitumor evaluation of a novel series of triaminotriazine derivatives Original Research Article

37

Synthesis and antitumor evaluation of benzoylphenylurea analogs

38

Synthesis and anti-tumor evaluation of new trisulfide derivatives

39

Synthesis and antitumor evaluation of novel 5-substituted-4-hydroxy-8-nitroquinazolines as EGFR signaling-targeted inhibitors Original Research Article

40

Synthesis and antitumor evaluation of novel monoindolyl-4-trifluoromethylpyridines and bisindolyl-4-trifluoromethylpyridines

41

Synthesis and antitumor evaluation of paclitaxel phosphonooxymethyl ethers: a novel class of water soluble paclitaxel pro-drugs

42

Synthesis and antitumor properties of 2,5-bis(3′-indolyl)thiophenes: Analogues of marine alkaloid nortopsentin

43

Synthesis and antitumor properties of a plasmalogen methyl ether analogue

44

Synthesis and antitumoral activities of marine ent-chromazonarol and related compounds

45

Synthesis and antitumoral activity of novel 3-(2-substituted-1,3,4-oxadiazol-5-yl) and 3-(5-substituted-1,2,4-triazol-3-yl) β-carboline derivatives Original Research Article

46

Synthesis and antitumoral evaluation of indole alkaloid analogues containing an hexahydropyrrolo[1′,2′,3′:1,9a,9]imidazo[1,2-a]indole skeleton Original Research Article

47

Synthesis and anti-tumor-promoting activity of glycoglycerolipid analogues lacking the glycerol backbone Original Research Article

48

Synthesis and antitumour activity of inositol phosphonate analogues

49

Synthesis and antitumour activity of new tiazofurin analogues bearing a 2,3-anhydro functionality in the furanose ring

50

Synthesis and antitumour activity of novel diterpenequinone salvicine and the analogs

51

Synthesis and antitumour activity of pyrene-linked pyrrolo [2,1-c] and benzodiazepine hybrids

52

Synthesis and antiviral activities of 1′-carbon-substituted 4′-thiothymidines Original Research Article

53

Synthesis and antiviral activities of N-9-oxypurine 1,3-Dioxolane and 1,3-oxathiolane nucleosides

54

Synthesis and antiviral activities of new acyclic and “double-headed” nucleoside analogues

55

Synthesis and antiviral activities of novel chiral cyanoacrylate derivatives with (E) configuration Original Research Article

56

Synthesis and antiviral activities of novel N-alkoxy-arylsulfonamide-based HIV protease inhibitors

57

Synthesis and antiviral activities of the major metabolites of the HIV protease inhibitor ABT-378 (Lopinavir)

58

Synthesis and antiviral activity against Coxsackie virus B3 of some novel benzimidazole derivatives

59

Synthesis and antiviral activity against tobacco mosaic virus and 3D-QSAR of α-substituted-1,2,3-thiadiazoleacetamides

60

Synthesis and Antiviral Activity of [2-[[4-[3-[(1-Methylethyl)amino]-2-Pyridyl]-1-Piperazinyl]Carbonyl]-1H-Indol-5-yl] (BHAP) Acylsphingosine HIV Reverse Transcriptase Inhibitors

61

Synthesis and antiviral activity of 2′-deoxy-2′-fluoro-2′-C-methyl purine nucleosides as inhibitors of hepatitis C virus RNA replication

62

Synthesis and antiviral activity of 2-deoxy-1,5-anhydro-D-mannitol nucleosides containing a pyrimidine base moiety

63

Synthesis and antiviral activity of 3′-C-branched-3′-deoxy analogues of adenosine

64

Synthesis and antiviral activity of 7-deazaneplanocin A against orthopoxviruses (vaccinia and cowpox virus)

65

Synthesis and antiviral activity of a new series of 4-isothiazolecarbonitriles Original Research Article

66

Synthesis and anti-viral activity of a series of d- and l-2′-deoxy-2′-fluororibonucleosides in the subgenomic HCV replicon system Original Research Article

67

Synthesis and anti-viral activity of a series of sesquiterpene lactones and analogues in the subgenomic HCV replicon system Original Research Article

68

Synthesis and antiviral activity of acyclovir-5′-(phenyl methoxy alaninyl) phosphate as a possible membrane-soluble nucleotide prodrug

69

Synthesis and antiviral activity of azoles obtained from carbohydrates

70

Synthesis and anti-viral activity of azolo-adamantanes against influenza A virus Original Research Article

71

Synthesis and antiviral activity of dihydroxycyclohexyl pyrimidine and purine carbocyclic nucleosides

72

Synthesis and antiviral activity of monobactams inhibiting the human cytomegalovirus protease Original Research Article

73

Synthesis and antiviral activity of new dimeric inhibitors against HIV-1 Original Research Article

74

Synthesis and antiviral activity of new phosphonobutoxypurines

75

Synthesis and antiviral activity of novel - and -2′-azido-2′,3′-dideoxyribofuranosyl-4′-thiopyrimidines and purines

76

Synthesis and antiviral activity of novel acyclic nucleosides in the 5-alkynyl- and 6-alkylfuro[2,3-d]pyrimidine series Original Research Article

77

Synthesis and antiviral activity of novel isodideoxy nucleosides with exocyclic methylene

78

Synthesis and antiviral activity of novel pyrazole derivatives containing oxime esters group Original Research Article

79

Synthesis and antiviral activity of P1′ arylsulfonamide azacyclic urea HIV protease inhibitors

80

Synthesis and antiviral activity of phosphonate derivatives of enantiomeric dihydro-2H-pyranyl nucleosides

81

Synthesis and antiviral activity of prodrugs of the nucleoside 1-[2′,3′-Dideoxy-3′-C-(hydroxymethyl)-β-d-erythropentofuranosyl] cytosine Original Research Article

82

Synthesis and antiviral activity of rigid acyclonucleotide analogs

83

Synthesis and antiviral activity of scopadulcic acids analogues

84

Synthesis and antiviral activity of some N-benzenesulphonylbenzimidazoles

85

Synthesis and antiviral effects of 2-heteroaryl substituted adenosine and 8-heteroaryl substituted guanosine derivatives Original Research Article

86

Synthesis and antiviral evaluation of 3-hydroxy-2-methylpyridin-4-one dideoxynucleoside derivatives

87

Synthesis and antiviral evaluation of 4′-hydroxymethyl-2′, 3′-dideoxy-3′-thianucleosides and their cyclic monophosphates

88

Synthesis and antiviral evaluation of acyclic azanucleosides developed from sulfanilamide as a lead structure Original Research Article

89

Synthesis and antiviral evaluation of benzimidazoles, quinoxalines and indoles from dehydroabietic acid Original Research Article

90

Synthesis and antiviral evaluation of enantiomeric 2′,3′-dideoxy- and 2′,3′-didehydro-2′,3′-dideoxy-4′-thionucleosides

91

Synthesis and antiviral evaluation of nucleic acid-based (NABTM) libraries

92

Synthesis and antiviral evaluation of some new pyrazole and fused pyrazolopyrimidine derivatives Original Research Article

93

Synthesis and Antiviral Properties of 1-Substituted 3-[ω-(4-Oxoquinazolin-4(3H)-yl)alkyl]uracil Derivatives

94

Synthesis and antiviral properties of aza-analogues of ganciclovir derived from 5,5-bis(hydroxymethyl)pyrrolidin-2-one

95

Synthesis and antiviral properties of some polyphenols related to Salvia genus

96

Synthesis and antiviral property of allophenylnorstatine-based HIV protease inhibitors incorporating d-cysteine derivatives as P2/P3 moieties

97

Synthesis and antiviral/antiproliferative activity of some N-sulphonylbenzimidazoles

98

Synthesis and antiviral/antitumor evaluation of 2-amino- and 2-carboxamido-3-arylsulfonylthiophenes and related compounds as a new class of diarylsulfones Original Research Article

99

Synthesis and apoptogenic activity of fluorinated ceramide and dihydroceramide analogues

100

Synthesis and appetite suppressant activity of 1-aryloxy-2-substituted aminomethyltetrahydronaphthalenes as conformationally rigid analogues of fluoxetine Original Research Article

101

Synthesis and application as polymer electrolyte of hyperbranched copolyethers derived from cationic ring-opening polymerization of 3-{2-[2-(2-methoxyethoxy)ethoxy]ethoxy}methyl- and 3-hydroxymethyl-3′-methyloxetane

102

Synthesis and application for overall water splitting of transition metal-mixed mesoporous Ta oxide

103

Synthesis and application in asymmetric copper(I)-catalyzed allylic oxidation of a new chiral 1,10-phenanthroline derived from pinene

104

Synthesis and application in high-pressure polymerization of a titanium complex with a linked cyclopentadienyl-phenoxide ligand

105

Synthesis and application in solar cell of poly(3-dodecylthiophene)/titanium dioxide nanocomposite Original Research Article

106

Synthesis and application in solar cell of poly(3-octylthiophene)/cadmium sulfide nanocomposite

107

Synthesis and application in SPPS of a stable amino acid isostere of palmitoyl cysteine

108

Synthesis and application of 2′-fluoro-substituted cap analogs

109

Synthesis and application of 2-styryl-6(7)-bromothiazolo[4,5-b]quinoxaline based fluorescent dye chromophores: Part 2

110

Synthesis and Application of 3,3-Diarylmethyl BINOLs

111

Synthesis and application of a carbamazepine-imprinted polymer for solid-phase extraction from urine and wastewater Original Research Article

112

Synthesis and application of a functionalized resin for flow injection/F AAS copper determination in waters

113

Synthesis and application of a functionalized resin in on-line system for copper preconcentration and determination in foods by flame atomic absorption spectrometry

114

Synthesis and application of a highly efficient tetraester calix[4]arene based resin for the removal of Pb2+ from aqueous environment Original Research Article

115

Synthesis and application of a macroporous boronate affinity monolithic column using a metal-organic gel as a porogenic template for the specific capture of glycoproteins

116

Synthesis and application of a new 2′,3′-isopropylidene guanosine substituted cap analog

117

Synthesis and application of a new functionalized resin for use in an on-line, solid phase extraction system for the determination of trace elements in waters and reference cereal materials by flame atomic absorption spectrometry

118

Synthesis and application of a new polystyrene-supported ruthenium carbene catalyst for alkene metathesis

119

Synthesis and application of a new selenoplatinum catalyst

120

Synthesis and Application of a Novel Fluorescent Reactive Dye Based on Fused Iminocoumarin on Cotton Fabric

121

Synthesis and application of a novel mesoporous zeolite L in the catalyst for the HDS of FCC gasoline Original Research Article

122

Synthesis and application of a novel single-isomer mono-6-deoxy-6-(3R,4R-dihydroxypyrrolidine)-β-cyclodextrin chloride as a chiral selector in capillary electrophoresis

123

Synthesis and application of a novel solid-phase microextraction adsorbent: Hollow fiber supported carbon nanotube reinforced sol–gel for determination of phenobarbital Original Research Article

124

Synthesis and application of a novel, crystalline phosphoramidite monomer with Thiol Terminus, suitable for the synthesis of DNA conjugates Original Research Article

125

Synthesis and application of a peroxidase-like molecularly imprinted polymer based on hemin for selective determination of serotonin in blood serum Original Research Article

126

Synthesis and application of a polyacrylate dispersant on the preparation of ultrafine ground calcium carbonate in a laboratory stirred media mill

127

Synthesis and application of a Sec2-containing oligopeptide for method evaluation purposes in selenium speciation

128

Synthesis and Application of a Sulfonated Carbon Catalyst for a Hydrolisis Reaction

129

Synthesis and application of a T-2 toxin imprinted polymer

130

Synthesis and application of Al and Sn doped TUD-1 mesoporous silica in removing methylene blue from water

131

Synthesis and application of Amberlite xad-4 functionalized with alizarin red-s for preconcentration and adsorption of rhodium (III)

132

Synthesis and Application of Aminmodified Fe3O4@MCM-41 Coreshell Magnetic Mesoporous for Effective Removal of pb^2+ ions from Aqueous Solutions and Optimization with Response Surface Methodology

133

Synthesis and application of amino-modified silicas containing albumin as hemoadsorbents for bilirubin adsorption

134

Synthesis and application of amphoteric starch graft polymer

135

Synthesis and application of amphoteric starch graft polymer

136

Synthesis and application of an alkali-clearable azo disperse dye containing a fluorosulfonyl group and analysis of its alkali-hydrolysis kinetics

137

Synthesis and application of an auxiliary group for chemical ligation at the X-gly site

138

Synthesis and application of an efficient calix[4]arene-based anion receptor bearing imidazole groups for Cr(VI) anionic species

139

Synthesis and application of an oxytetracycline imprinted polymer for the solid-phase extraction of tetracycline antibiotics Original Research Article

140

Synthesis and application of atropisomeric dihydrobenzofuran-based bisphosphine (BICMAP)

141

Synthesis and Application of Benzotriazols as UVAbsorbers

142

Synthesis and Application of Benzotriazols as UVAbsorbers

143

Synthesis and application of benzyl-TMS derivatives as bench stable benzyl anion equivalents

144

Synthesis and Application of Bis[1,2-(4-aryl-2-alkyl-1H- inden-1-yl)]Ethane as an Efficient`Ligand for Preparation of Olefin Polymerization Catalysts

145

Synthesis and application of calcium sulphate pigment for paper coating: Potential and prospects

146

Synthesis and application of cationic starch graft polymer by using the complex initiation system

147

Synthesis and application of cationised cellulose for removal of Cr(VI) from acid mine-drainage contaminated water

148

Synthesis and application of chelating resins based on polyacrylonitrilediethylenetriamine for metal ions removal

149

Synthesis and application of chiral hydrobenzoin

150

Synthesis and application of cinnamate-functionalized rubber for the preparation of UV-curable films

151

Synthesis and application of CNT-supported MoO3-K2O nanocatalyst using microemulsion technique: role of nanoparticle size on catalyst activity and selectivity in higher alcohol synthesis

152

Synthesis and application of conducting graft copolymer with viable processability

153

Synthesis and application of crown ether tagged triarylphosphines

154

Synthesis and application of dehydroabietylisothiocyante as a new chiral derivatizing agent for the enantiomeric separation of chiral compounds by capillary electrophoretic Original Research Article

155

Synthesis and application of direct black dyes containing 4,4-diaminodiphenyl sulfonamide

156

Synthesis and application of DNA-templated silver nanowires for ammonia gas sensing

157

Synthesis and application of double metal MXenes: A review

158

Synthesis and application of doxorubicin-loaded silica gels as solid materials for spectral analysis

159

Synthesis and application of epoxy starch derivatives

160

Synthesis and application of epoxy starch derivatives

161

Synthesis and Application of Fe3O4@Au Composite Nanoparticles as Magnetic Resonance/Computed Tomography Dual‑Modality Contrast Agent

162

Synthesis and application of fluorescently labeled phthalic anhydride (PA) functionalized polymers by ATRP

163

Synthesis and application of functional polyethylene graft copolymers by atom transfer radical polymerization

164

Synthesis and application of functionally diverse 2,6,9-trisubstituted purine libraries as CDK inhibitors Original Research Article

165

Synthesis and application of gold-carbon hybrids as catalysts for the hydroamination of alkynes Original Research Article

166

Synthesis and application of H-Bonded cross-linking polymers containing a conjugated pyridyl H-Acceptor side-chain polymer and various carbazole-based H-Donor dyes bearing symmetrical cyanoacrylic acids for organic solar cells

167

Synthesis and Application of Heterocyclic as ultraviolet Absorbers

168

Synthesis and Application of Hydrogels for Oil-Water Separation

169

Synthesis and application of hydroxyapatite/polylactide composite biomaterial

170

Synthesis and application of hypercrosslinked polymers with weak cation-exchange character for the selective extraction of basic pharmaceuticals from complex environmental water samples

171

Synthesis and application of imprinted polyvinylimidazole-silica hybrid copolymer for Pb2+ determination by flow-injection thermospray flame furnace atomic absorption spectrometry Original Research Article

172

Synthesis and Application of Inorganic Nanoparticles as Lubricant Components – a Review

173

Synthesis and application of ionic liquid matrices (ILMs) for effective pathogenic bacteria analysis in matrix assisted laser desorption/ionization (MALDI-MS) Original Research Article

174

Synthesis and application of ion-imprinted polymer nanoparticles for the extraction and preconcentration of zinc ions

175

Synthesis and Application of Iron Oxide/Silica Gel Nanocomposite for Removal of Sulfur Dyes from Aqueous Solutions

176

synthesis and application of iron oxide/silica gel nanocomposite for removal of sulfur dyes from aqueous solutions

177

Synthesis and Application of Iron Oxide/Silica Gel Nanocomposite for Removal of Sulfur Dyes from Aqueous Solutions

178

Synthesis and Application of Jatropha Oil based Polyurethane as Paint Coating Material

179

Synthesis and application of layered double hydroxide-hosted catalysts for stereoselective epoxidation using molecular oxygen or air

180

Synthesis and application of lead telluride nanoparticles for degrediation of organic pollution

181

Synthesis and application of L-proline and R-phenylglycine derived organocatalysts for direct asymmetric Michael addition of cyclohexanone to nitroalkenes

182

Synthesis and application of magnesium oxide nanospheres with high surface area

183

Synthesis and Application of Magnetic Fe3O4Walnut Sawdust Nanocomposite for Removal of Lead from Water

184

Synthesis and Application of Magnetic Nanoadsorbent in Removal of Toxic Metals from Aqueous Solution

185

Synthesis and application of magnetite dextran-spermine nanoparticles in breast cancer hyperthermia

186

Synthesis and application of metal complex dyes derived from5-arylazo-4-hydroxy-2-phenylpyridazin-3-one

187

Synthesis and application of metal complex dyes derived from5-arylazo-4-hydroxy-2-phenylpyridazin-3-one

188

Synthesis and application of micro-mesoporous SBA-3 with 1,2-bis(triethoxysilyl)ethane as secondary silica source

189

Synthesis and application of modified magnetic nanoparticles for removal of Cyanide from aqueous solutions

190

Synthesis and application of modified vegetable oils in water-repellent finishing of cotton fabrics

191

Synthesis and application of modified vegetable oils in water-repellent finishing of cotton fabrics

192

Synthesis and application of moisture-stable methallylsilanated phosphorylcholine as a surface modifier

193

Synthesis and application of molecularly imprinted poly(methacrylic acid)–silica hybrid composite material for selective solid-phase extraction and high-performance liquid chromatography determination of oxytetracycline residues in milk

194

Synthesis and application of molecularly imprinted polymer on selective solid-phase extraction for the determination of monosulfuron residue in soil

195

Synthesis and application of molecularly imprinted polymer on selective solid-phase extraction for the determination of monosulfuron residue in soil

196

Synthesis and application of mono-2A-azido-2A-deoxyperphenylcarbamoylated β-cyclodextrin and mono-2A-azido-2A-deoxyperacetylated β-cyclodextrin as chiral stationary phases for high-performance liquid chromatography

197

Synthesis and application of mono-6-(3-methylimidazolium)-6-deoxyperphenylcarbamoyl-β-cyclodextrin chloride as chiral stationary phases for high-performance liquid chromatography and supercritical fluid chromatography

198

Synthesis and application of mono-6-ammonium-6-deoxy-β-cyclodextrin chloride as chiral selector for capillary electrophoresis

199

Synthesis and Application of Monofunctional ReactiveDyes Based on 3-(4-amino phenyl)-5-Benzylidene-2SubstitutedPhenyl-3, 5-Dihydro-Irnidazol-4-0ne

200

Synthesis and application of monoterpene-based chiral aminodiols

201

Synthesis and application of multi-walled carbon nanotubes–molecularly imprinted sol–gel composite material for on-line solid-phase extraction and high-performance liquid chromatography determination of trace Sudan IV Original Research Article

202

Synthesis and application of nano-pore size ion imprinted polymer for solid phase extraction and determination of zinc in different matrices

203

Synthesis and application of new fullerene derivative

204

Synthesis and Application of New Gadolinium-Porphyrins as Potential MR Imaging Contrast Agents for Cancer Detection in Nude Mice

205

Synthesis and Application of New Oxidant bis(banzyltriphenylphosphonium) peroxodisulfate on Oxidation of Benzylhalides to Corresponding Benzylaldehyde Compounds

206

Synthesis and Application of New Oxidant bis(banzyltriphenylphosphonium) peroxodisulfate on Oxidation of Benzylhalides to Corresponding Benzylaldehyde Compounds

207

Synthesis and Application of New Quinoline as Hydrochloric Acid Corrosion Inhibitor of Carbon Steel

208

Synthesis and application of new sizing and finishing additives based on carboxymethyl cellulose

209

Synthesis and application of new temperature-responsive hydrogels based on carboxymethyl and hydroxyethyl cellulose derivatives for the functional finishing of cotton knitwear

210

Synthesis and application of novel ionic phosphine ligands with a cobaltocenium backbone

211

Synthesis and Application of Novel Modified Magnetic Nanocomposite for Solid Phase Extraction of Thallium(I) Ions

212

Synthesis and application of ortho-palladated complex of (4-phenylbenzoylmethylene)triphenylphosphorane as a highly active catalyst in the Suzuki cross-coupling reaction

213

Synthesis and application of poly(ethylene glycol)–cholesterol (Chol–PEGm) conjugates in physicochemical characterization of nonionic surfactant vesicles

214

Synthesis and Application of Polyacrylamide/Cellulose Gel/Fuller’s Earth Composite for Removal of Methylene Blue from Water

215

Synthesis and Application of Polyaniline/Multi Walled Carbon Nanotube Nanocomposite for Electrochemical Determination of Folic acid

216

Synthesis and application of polymer-supported N-sulfonylated aminoalcohols as enantioselective catalysts

217

Synthesis and application of polypyrrole/carrageenan nano-bio composite as a cathode catalyst in microbial fuel cells

218

Synthesis and application of polytetrahydrofuran-grafted polystyrene (PS–PTHF) resin supports for organic synthesis

219

Synthesis and application of proline based organocatalyst for highly enantioselective aldol reaction by hydrogen bonding

220

Synthesis and Application of Ruthenium(II) Tricarboxyterpyridyl Complex with a Nitrogen Chelete Ligand for Solar Cells Based on Nanocrystalline TiO2 Films

221

Synthesis and application of spherical macroporous epoxy-polyamide chelating resin for preconcentration and separation of trace Ga(III), In(III), Bi(III), V(V), Cr(III), and Ti(IV) from solution samples

222

Synthesis and application of starch-graft-poly(AM-co-AMPS) by using a complex initiation system of CS-APS

223

Synthesis and application of styrene/4-hydroxystyrene gradient copolymers made by controlled radical polymerization: Compatibilization of immiscible polymer blends via hydrogen-bonding effects

224

Synthesis and application of terpolymer scale inhibitor in the presence of β-cyclodextrins

225

Synthesis and application of the drilling mud additive in the presence of surfactants

226

Synthesis and application of the solar cell of poly(3-hexylthiophene)/Fe N/titanium dioxide nanocomposite material Original Research Article

227

Synthesis and application of Ti-incorporated mesoporous silicate in deep oxidesulfurization of DBT from liquid fuel

228

Synthesis and Application of TiO2/SWCNTs/Pt Nanocomposites as a Good Photocatalyst for Hydrogen Production

229

Synthesis and Application of Two Organic Dyes Based on Indoline in Dye Sensitized Solar Cells

230

Synthesis and Application of Two Organic Dyes for Dye-Sensitized Solar Cells

231

Synthesis and application of weight function for edge cracked semicircular disk (ECSD)

232

Synthesis and application of α-d-mannosyl clusters as photoaffinity ligands for mannose-binding proteins: Concanavalin A as a model receptor

233

Synthesis and application to asymmetric allylic amination of substituted monodonor diazaphospholidine ligands

234

Synthesis and Applicationof New Fluorescein Analogues

235

Synthesis and Applicationof New Fluorescein Analogues

236

Synthesis and applications of a chiral-oxygenated 3-chloro-3,6-dihydro-2H-pyran obtained under Overman rearrangement conditions

237

Synthesis and applications of a deep, asymmetric cavitand on a solid support

238

Synthesis and applications of a new palladacycle as a high active catalyst in the Suzuki couplings

239

Synthesis and Applications of beta-Aminocarboxylic Acids Containing a Cyclopropane Ring

240

Synthesis and applications of bis(perfluorodecalin-1-carbonyl) peroxide

241

Synthesis and applications of C2-symmetric guanidine bases

242

Synthesis and applications of chiral bis-THF in asymmetric synthesis

243

SYNTHESIS AND APPLICATIONS OF COUMARIN

244

Synthesis and Applications of Cross-linked Poly(N-bromomaleimide) in Oxidation of Various Organic Compounds

245

Synthesis and applications of diethylstilbestrol-based molecularly imprinted polymer-coated hollow fiber tube Original Research Article

246

Synthesis and applications of Fe3O4-diisopropylaminoacetamide as a versatile and reusable magnetic nanoparticle supported N,N-diisopropylethylamine equivalent

247

Synthesis and applications of fluorinated nucleoside analogues

248

Synthesis and applications of fluoroalkyl end-capped cooligomers having fullerene and mixed fullerenes in the main chain

249

Synthesis and applications of fulleropyrrolidines

250

Synthesis and applications of heterobifunctional poly(ethylene oxide) oligomers

251

Synthesis and applications of hyperbranched polyesters—preparation and characterization of crystalline silver nanoparticles

252

Synthesis and applications of hyperbranched polymers

253

Synthesis and applications of non-racemic cyanohydrins and α-amino nitriles

254

Synthesis and applications of novel acceptor–donor–acceptor organic dyes with dithienopyrrole- and fluorene-cores for dye-sensitized solar cells

255

Synthesis and applications of one-dimensional nano-structured polyaniline: An overview

256

Synthesis and applications of one-dimensional semiconductors

257

Synthesis and applications of optically active metallacycles derived from primary amines

258

Synthesis and Applications of Poly(N-vinylimidazole) Grafted Silica-containing Palladium Nanoparticles as a New Re-cyclable Catalyst for Heck, Sonogashira and Suzuki Coupling Reactions

259

Synthesis and applications of polysiloxanes containing photocrosslinkable oxaalkylene styrenyl groups

260

Synthesis and applications of propargyl pentafluorophenyl carbonate for peptide synthesis

261

Synthesis and applications of sulfonated polyaniline

262

Synthesis and applications of sulfur-substituted cis-hexahydro-2-quinolinones

263

Synthesis and applications of surface-grafted Th(IV)-imprinted polymers for selective solid-phase extraction of thorium(IV) Original Research Article

264

Synthesis and applications of surfactants containing fluorine

265

Synthesis and applications of tert-alkoxysiloxane linkers in solid-phase chemistry

266

Synthesis and applications of tetrathiafulvalenes and ferrocene-tetrathiafulvalenes and related compounds

267

Synthesis and applications of triblock and multiblock copolymers using telechelic oligopropylene

268

Synthesis and applications of vegetable oil-based fluorocarbon water repellent agents on cotton fabrics

269

Synthesis and aqueous solution behavior of phosphonate-functionalized chitosans

270

Synthesis and aqueous solution characterization of amphiphilic diblock copolymers containing carbazole

271

Synthesis and aqueous solution characterization of catalytically active homopolymers, block copolymers and networks containing imidazole

272

Synthesis and aqueous solution characterization of novel diblock polyampholytes containing imidazole

273

Synthesis and aqueous solution properties of near-monodisperse tertiary amine methacrylate homopolymers and diblock copolymers

274

Synthesis and aqueous solution properties of PAMAM dendron surfactants bearing a quaternary ammonium focal group and sugar terminal groups

275

Synthesis and Aromatic Diamine Intercalation of Graphene Oxide to Tailor the Electrochemical Properties

276

Synthesis and aromatic nucleophilic N–N, N–S and N–O exchange reactions of N,N-dimethyl-2-trifluoroacetyl-1-naphthylamine

277

Synthesis and arylation of unprotected sulfonimidamides

278

Synthesis and assay of isoquinoline derivatives as HIV-1 Tat–TAR interaction inhibitors

279

Synthesis and assembly of Bi2S3 nanoparticles at the water–toluene interface

280

Synthesis and assembly of catalytically active platinum-doped polymer nanocomposites at the liquid/liquid interface

281

Synthesis and assembly of oligoaniline for hierarchical structures within stable and mild acid system

282

Synthesis and assembly of zinc hydroxide sulfate large flakes: Application in gas sensor based on a novel surface mount technology

283

Synthesis and assessment of date palm genetic diversity studies

284

Synthesis and assessment of La0.8Sr0.2ScyMn1−yO3−δ as cathodes for solid-oxide fuel cells on scandium-stabilized zirconia electrolyte

285

Synthesis and assessment of new cyclopenta-2,4-dienone derivatives for energy storage applications

286

Synthesis and assessment of new cyclopenta-2,4-dienone derivatives for energy storage applications

287

Synthesis and assessment of the effect of monomer feed ratio and Lewis acids on copolymerization of butyl methacrylate/1-octene

288

Synthesis and association of Ag(0) nanoparticles in aqueous Pluronic F127 triblock copolymer solutions

289

Synthesis and association properties of thermoresponsive and permanently cationic charged block copolymers

290

Synthesis and asymmetric catalytic activities of chiral organogallium and indium complexes with ephedrine derivatives as ligands. The crystal structure of [(1R, 2S)-(Me2Ga-μ-OCH(C6H5)CH(CH3)-μ-NHCH3)]2

291

Synthesis and asymmetric catalytic application of chiral imidazolium–phosphines derived from (1R,2R)-trans-diaminocyclohexane

292

Synthesis and asymmetric hydrogenation of 3,5-dioxoheptanedioates. Preparation of enantiomerically pure substituted δ-valerolactones

293

Synthesis and atom-scale microstructure of Ba6Mn5O16 Original Research Article

294

Synthesis and atropisomerism of 2,2′-ortho disubstituted biphenyls

295

Synthesis and ATRP of novel fluorinated aromatic monomer with pendant sulfonate group

296

Synthesis and Autoradiographic Evaluation of a Novel High-Affinity Tc-99m Ligand for the 5-HT2A Receptor

297

Synthesis and autoradiographic localization of muscarinic cholinergic antagonist (+)N-[11C]methyl-3-piperidyl benzilate as a potent radioligand for positron emission tomography

298

Synthesis and autoradiographic localization of the dopamine D-1 agonists [11C]SKF 75670 and [11C]SKF 82957 as potential PET radioligands

299

Synthesis and axial ligation behaviour of sterically hindered Zn(II)–porphyrin liquid crystals

300

Synthesis and Bacterial Evaluation of The V(IV), Cr(III), Fe(III) and Co(II) Ions Complexes with Mixed Ligands (2-hydroxybenzaldine)-4- Aminoantipyrine and 8-Hydroxyquinoline

301

Synthesis and bacterial expression of a gene encoding the heme domain of assimilatory nitrate reductase

302

Synthesis and bactericidal ability of Ag/TiO2 composite films deposited on titanium plate

303

Synthesis and Bactericidal Efficacy of Novel Dendrimers

304

Synthesis and barrier properties of poly(vinylidene chloride-co-acrylonitrile)/SiO2 hybrid composites by sol–gel process

305

Synthesis and baseline testing of a digital pulse-width-modulated clutch

306

Synthesis and basic properties of tetrathieno[2,3-a:3′,2′-c:2″,3″-f:3‴,2‴-h]naphthalene: a new π-conjugated system obtained by photoinduced electrocyclization–dehydrogenation reactions of tetra(3-thienyl)ethene

307

Synthesis and behavior evaluation of a relative permeability modifier

308

Synthesis and Behavior of α-Iminocarboxyamide Nickel and Zirconium Catalysts Towards Olefin Polymerization

309

Synthesis and benzodiazepine receptor (ω receptor) affinities of 3-substituted derivatives of pyrrolo[2,3-c]pyridine-5-carboxylate, a novel class of ω1 selective ligands Original Research Article

310

Synthesis and binding activity of endomorphin-1 analogues containing β-amino acids

311

Synthesis and binding affinities of 2β-(3-iodoallyloxycarbonyl)-3β-(4-substituted-aryl)tropane analogues as ligands for the dopamine transporter studies

312

Synthesis and binding affinities of 4-diarylaminotropanes, a new class of delta opioid agonists

313

Synthesis and binding affinities of methylvesamicol analogs for the acetylcholine transporter and sigma receptor Original Research Article

314

Synthesis and binding affinity of 2,3,3a,4,9,9a-hexahydro-9,4-(iminomethano)-1H-benz[f]indenes. Ligands for the PCP site of the NMDA receptor

315

Synthesis and binding affinity of neuropeptide Y at opiate receptors

316

Synthesis and binding affinity of new muscarinic ligands structurally related to oxotremorine

317

Synthesis and binding affinity of new pyrazole and isoxazole derivatives as potential atypical antipsychotics

318

Synthesis and binding affinity of novel 3-aminoethyl-1-tetralones, potential atypical antipsychotics

319

Synthesis and binding analysis of unique AG2 pentasaccharide to human Siglec-2 using NMR techniques Original Research Article

320

Synthesis and binding behavior of a Zn(II)-porphyrin having calix[5]arene cap

321

Synthesis and binding behaviors of monomethyl cucurbit[6]uril

322

Synthesis and Binding Characteristics of N-(l-Naphthyl)-N(3-[125 I]-iodophenyl)-N-methylguanidine ([125I]-CNS 1261): A Potential SPECT Agent for Imaging NMDA Receptor activation

323

Synthesis and binding mode of heterocyclic analogues of suramin inhibiting the human basic fibroblast growth factor Original Research Article

324

Synthesis and binding of stable bisubstrate ligands for phosphoglycerate kinase

325

Synthesis and binding properties of a macrocycle with two binding subcavities

326

Synthesis and binding properties of carboxylphenyl-modified calix[4]arenes and cytochrome c

327

Synthesis and binding properties of cyclodextrin trimers

328

Synthesis and binding properties of cyclopentane analogues of myo-inositol 1,4,5-tris(phosphate) Original Research Article

329

Synthesis and binding properties of myo-inositol 4,5,6-tris(phosphate) an analogue of myo-inositol 1,4,5-tris(phosphate). Correlation with the ionization state of the molecules

330

Synthesis and binding properties of novel selective 5-HT3 receptor ligands Original Research Article

331

Synthesis and binding properties of oligodeoxynucleotides containing phenylphosphon(othio)ate linkages Original Research Article

332

Synthesis and binding properties of perylene-oligo-2′-deoxyribonucleotide conjugates

333

Synthesis and binding properties of photoactivable biotin-conjugated verapamil derivatives for the study of P-170 glycoprotein Original Research Article

334

Synthesis and binding selectivity of 7- and 15-decylbenzolactone-V8 for the C1 domains of protein kinase C isozymes

335

Synthesis and binding studies of 2-O- and 11-O-substituted N-alkylnoraporphines

336

Synthesis and binding studies of a 1-alkyl-3,6-diamino-4-quinolone based receptor for N-acylated dipeptides

337

Synthesis and binding studies of carboxylate binding pocket analogs of vancomycin

338

Synthesis and binding studies of multiple calix[4]arenes

339

Synthesis and binding studies of new bis-calix[4]arenes containing aromatic and heteroaromatic units

340

Synthesis and binding studies of novel bisthiacalix[4]arenes with diimime linkages

341

Synthesis and binding studies of novel thiacalixpodands and bisthiacalixarenes having O,O″-dialkylated thiacalix[4]arene unit(s) of 1,3-alternate conformation

342

Synthesis and binding studies of some epibatidine analogues

343

Synthesis and binding to plant lectins of sulfur-containing analogues of βGal1,3αGalNAc (T-antigen)

344

Synthesis and binding with BSA of a new gemini surfactant

345

Synthesis and bioactive properties of macroporous nanoscale SiO2–CaO–P2O5 bioactive glass

346

Synthesis and bioactivities of 6,7,8-trimethoxy-N-aryl-4-aminoquinazoline derivatives Original Research Article

347

Synthesis and bioactivities of heterocyclic lipids as PAF antagonists. 1

348

Synthesis and bioactivities of heterocyclic lipids as PAF antagonists. 2

349

Synthesis and bioactivities of nitronyl nitroxide and RGD containing pseudopeptides

350

Synthesis and bioactivities of novel 4,5,6,7-Tetrahydrothieno[2,3-c]pyridines as inhibitors of tumor necrosis factor-α (TNF-α) production

351

Synthesis and bioactivities of novel 5,6-Bis(4-methoxyphenyl)-2H-pyridazin-3-one derivatives: inhibitors of interleukin-1 beta (IL-1β) production

352

Synthesis and bioactivities of novel bicyclic thiophenes and 4,5,6,7-tetrahydrothieno[2,3-c]pyridines as inhibitors of tumor necrosis factor-α (TNF-α) production

353

Synthesis and bioactivities of novel piperidylpyrimidine derivatives: inhibitors of tumor necrosis factor-alpha production

354

Synthesis and bioactivities of novel pyridazine derivatives: inhibitors of interleukin-1 beta (IL-1β) production

355

Synthesis and bioactivities of paclitaxel analogs with a cyclopropanated side-chain

356

Synthesis and bioactivities of poly(ethylene glycol)¯chitosan hybrids

357

Synthesis and bioactivities of two multiple antigen peptides as potential vaccine against schistosoma

358

Synthesis and bioactivity of (±)-tetrahydrohaliclonacyclamine A

359

Synthesis and bioactivity of 2,4-diacyl analogues of paclitaxel Original Research Article

360

Synthesis and bioactivity of 2-cyanoacrylates containing a trifluoromethylphenyl moiety

361

Synthesis and bioactivity of 4,10-dimethyl-pyridino[2,3-h]quinolin-2(1H)-one-9-carboxylic acid and its esters Original Research Article

362

Synthesis and bioactivity of 4-alkyl(aryl)thioquinazoline derivatives

363

Synthesis and bioactivity of 5-(1-aryl-1H-tetrazol-5-ylsulfanylmethyl)-N-xylopyranosyl-1,3,4-oxa(thia)diazol-2-amines Original Research Article

364

Synthesis and Bioactivity of a Cyclopolypeptide from Caribbean Marine Sponge

365

Synthesis and bioactivity of fluorescence- and biotin-labeled lipid A analogues for investigation of recognition mechanism in innate immunity

366

Synthesis and bioactivity of fluorine compounds containing isoxazolylamino and phosphonate groups

367

Synthesis and bioactivity of highly ordered TiO2 nanotube arrays

368

Synthesis and bioactivity of new antineoplastic terpenylquinones

369

Synthesis and bioactivity of novel (3-chloro-5-(trifluoromethyl)pyridin-2-yloxy)phenyl containing acrylate and acrylonitrile derivatives

370

Synthesis and bioactivity of novel methyl 6-deoxy-6-(N′-alkyl/aryl-N″-benzothiazol-2-yl)guanidino-α-d-glucopyranosides Original Research Article

371

Synthesis and bioactivity of photolabile sirolimus (rapamycin) analogs

372

Synthesis and bioactivity of porous Ti alloy prepared by foaming with TiH2

373

Synthesis and bioactivity of α-galactosylceramide analogues bearing an aryl group within the fatty amide chain

374

Synthesis and bioanalytical applications of specific-shaped metallic nanostructures: A review Review Article

375

Synthesis and bio-applications of carbohydrate–gold nanoconjugates with nanoparticle and nanolayer forms

376

Synthesis and bioassay evaluation of 1-(4-substitutedideneaminooxymethyl)-phenyl-3-(2,6-difluorobenzoyl)ureas Original Research Article

377

Synthesis and bioassay of 4-ipomeanol analogs as potential chemopreventive agents against 4-(methylnitrosamino)-1-(3-pyridyl)-1-butanone (NNK)-induced tumorigenicity in A/J mice

378

Synthesis and bioassay of a protein tyrosine phosphatase inhibitor, dephostatin

379

Synthesis and biochemical activity of novel amidine derivatives as m1 muscarinic receptor agonists Original Research Article

380

Synthesis and biochemical application of 2′-O-methyl-3′-thioguanosine as a probe to explore group I intron catalysis Original Research Article

381

Synthesis and biochemical applications of a solid cyclic nitrone spin trap: a relatively superior trap for detecting superoxide anions and glutathiyl radicals

382

Synthesis and Biochemical effects of magnetite nanoparticle by surfactantfree electrochemical method in an aqueous system:the current density effect

383

Synthesis and biochemical evaluation of a range of potent benzyl imidazole-based compounds as potential inhibitors of the enzyme complex 17α-hydroxylase/17,20-lyase (P45017α)

384

Synthesis and biochemical evaluation of des-vinyl secologanin aglycones with alternate stereochemistry

385

Synthesis and biochemical evaluation of RNA containing an intrahelical disulfide crosslink Original Research Article

386

Synthesis and biochemical investigation of scyphostatin analogues as inhibitors of neutral sphingomyelinase Original Research Article

387

Synthesis and Biochemical Properties of Cyanuric Acid Nucleoside-Containing DNA Oligomers

388

Synthesis and biochemical properties of E-ring modified luotonin A derivatives

389

Synthesis and biochemical properties of oligodeoxynucleotides acylated by the chemically stable 2-(trimethylsilyl)benzoyl (TMSBz) group at the 5′ or 3′ terminus

390

Synthesis and biochemical properties of Z- and E-4,5-dehydrodethiobiotin Original Research Article

391

Synthesis and biocidal activity of some new 2-amino-4,6-diarylsubstituted-pyrimidines

392

Synthesis and biocompatibility evaluation of cellulose/hydroxyapatite nanocomposite scaffold in 1-n-allyl-3-methylimidazolium chloride

393

Synthesis and biocompatibility of a novel silicone hydrogel containing phosphorylcholine

394

Synthesis and biocompatibility of anionic polyurethane nanoparticles coated with adsorbed chitosan

395

Synthesis and biodegradability of starch-g-ethyl methacrylate/ sodium acrylate/sodium silicate superabsorbing composite

396

Synthesis and biodegradation of arabinogalactan sponges prepared by reductive amination

397

Synthesis and biodegradation studies of 1,3-propanediol based aliphatic poly(ester carbonate)s

398

Synthesis and biodegradation studies of new copolymers based on sucrose derivatives and styrene

399

Synthesis and Biodistribution of (R,S)-[O-Methyl-11C]-1-[3-(5-Methoxy-1,2,3,4-tetrahydro-1-naphtalenyl)propyl]-4-Phenylpiperazine (PNU-157760), A Putative Radioligand for 5-HT1AReceptors

400

Synthesis and biodistribution of [11C]A-836339, a new potential radioligand for PET imaging of cannabinoid type 2 receptors (CB2) Original Research Article

401

Synthesis and biodistribution of [11C]procaterol, a β2-adrenoceptor agonist for positron emission tomography

402

Synthesis and biodistribution of [11C]R116301, a promising PET ligand for central NK1 receptors Original Research Article

403

Synthesis and biodistribution of 2-[123I]iodomelatonin in normal mice

404

Synthesis and biodistribution of 34mCl-labeled 2-chloro-2-deoxy-d-glucose: A major impurity in [18F]FDG injection

405

Synthesis and biodistribution of 8-iodo-11-(4-methylpiperazino)-5H-dibenzo[b,e][1,4]-diazepine: Iozapine

406

Synthesis and biodistribution of 99mTc-carbonyltechnetium-labeled fatty acids

407

Synthesis and biodistribution of a new 99mTc nitrido complex as a potential myocardial and cerebral imaging agent

408

Synthesis and biodistribution of a new 99mTc nitrido complex for brain imaging

409

Synthesis and biodistribution of a novel 99mTcN complex of ciprofloxacin dithiocarbamate as a potential agent for infection imaging

410

Synthesis and biodistribution of new radiolabeled high-affinity choline transporter inhibitors [11C]hemicholinium-3 and [18F]hemicholinium-3

411

Synthesis and Biodistribution of R- and S-lsomers of [18 F]-Fluoropropranolol, a Lipophilic Ligand for the beta-Adrenergic Receptor

412

Synthesis and biodistribution of six novel 99mTc complexes of 2-hydroxybenzaldehyde-amino acid Schiff bases

413

Synthesis and biodistribution of two novel 99mTc( SNN/S) “3+1” mixed ligand complexes as potential brain perfusion agents

414

Synthesis and biodistribution study of a chlorotoxin derivative peptide labeled with 131- iodine for tumor therapy

415

Synthesis and bioevaluation of 22-hydroxyacuminatine analogs

416

Synthesis and bioevaluation of hybrid 4-aminoquinoline triazines as a new class of antimalarial agents

417

Synthesis and Bioevaluation of Iodine-131 Directly Labeled Cyclic RGD-PEGylated Gold Nanorods for Tumor-Targeted Imaging

418

Synthesis and bioevaluation of N-(arylalkyl)-homospermidine conjugates

419

Synthesis and biologic studies of iodinated (125I/127I) ethidium

420

Synthesis and biological activation of an ethylene glycol-linked amino acid conjugate of cyclic cidofovir

421

Synthesis and biological activities of [N-MeLeu5] didemnin B

422

Synthesis and biological activities of 1-pyridylisoquinoline and 1-pyridyldihydroisoquinoline derivatives as PDE4 inhibitors

423

Synthesis and biological activities of 2′-deoxy-2′-fluoro-4′-thioarabinofuranosylpyrimidine and -purine nucleosides Original Research Article

424

Synthesis and biological activities of 2-methyl-4-N-2́-cyanoethyl-N-substituted benzaldehydes and their derivatives

425

Synthesis and biological activities of 2-oxocycloalkylsulfonamides Original Research Article

426

Synthesis and biological activities of 3-polyamino-5β-cholane-7α,24-diols

427

Synthesis and biological activities of 5′-ethylenic and acetylenic modified l-nucleosides and isonucleosides

428

Synthesis and biological activities of 7-aza rebeccamycin analogues bearing the sugar moiety on the nitrogen of the pyridine ring Original Research Article

429

Synthesis and biological activities of a novel class of azole-containing antifungal agents

430

Synthesis and biological activities of an α-methyl and a β-methyl carbapenem and the corresponding unsubstituted compound

431

Synthesis and biological activities of analogs of d-glucosyl-l-tyrosine, a humoral factor that stimulates transcription of the acyl-CoA binding protein in the pheromone gland of the Silkmoth, Bombyx mori Original Research Article

432

Synthesis and biological activities of aryl-ether-, biaryl-, and fluorene-aspartic acid and diaminopropionic acid analogs as potent inhibitors of the high-affinity glutamate transporter EAAT-2

433

Synthesis and biological activities of camphor-based non-peptide growth hormone secretagogues

434

Synthesis and biological activities of flavolipids

435

Synthesis and biological activities of fluorinated 10-hydroxycamptothecin and SN38

436

Synthesis and biological activities of fluorinated chalcone derivatives Original Research Article

437

Synthesis and biological activities of fluorine-containing N,N′-diphenylcarbamimidothioates

438

Synthesis and biological activities of glycosphingolipid analogues from marine sponge Aplysinella rhax

439

Synthesis and biological activities of hapalosin derivatives with modification at the C12 position

440

Synthesis and biological activities of hydroxyl-protected fluorine-containing 4,4-dihydroxylmethyl-2-aryl-iminothiazolidines

441

Synthesis and biological activities of isogranulatimide analogues Original Research Article

442

Synthesis and Biological Activities of Lipid A Analogs Possessing (beta)-Glycosidic Linkage at 1-Position

443

Synthesis and biological activities of lipid A-type pyrancarboxylic acid derivatives

444

Synthesis and biological activities of methylenebis-4H-1,2,4-triazole derivatives

445

Synthesis and biological activities of N-(1,2,4-triazole-4-yl)-N′-(fluorine-containing-phenyl)carbamimidothioates

446

Synthesis and biological activities of NB-506 analogues modified at the glucose group

447

Synthesis and biological activities of NB-506 analogues: Effects of the positions of two hydroxyl groups at the indole rings

448

Synthesis and biological activities of new 1H-1,2,4-triazole derivatives containing ferrocenyl moiety

449

Synthesis and biological activities of new 1α,25-dihydroxy-19-norvitamin D3 analogs with modifications in both the A-ring and the side chain Original Research Article

450

Synthesis and biological activities of new conformationally fixed analogues of (−)-indolactam-V, the core structure of tumor-promoting teleocidins

451

Synthesis and biological activities of new heterocyclic aromatic retinoids

452

Synthesis and Biological Activities of Nickel(II) and Cadmium(II) Complexes of Chlorohydroxyacetophenone-nitrobenzoylhydrazone: Mechanism for Formation of the Nickel(II) complex

453

Synthesis and biological activities of novel 17-aminogeldanamycin derivatives Original Research Article

454

Synthesis and biological activities of novel 4″-alkylidene avermectin derivatives

455

Synthesis and biological activities of novel antiallergic agents with 5-lipoxygenase inhibiting action Original Research Article

456

Synthesis and biological activities of novel aryl indole-2-carboxylic acid analogs as PPARγ partial agonists

457

Synthesis and biological activities of novel dexibuprofen tetraacetylriboflavin conjugates

458

Synthesis and biological activities of novel dialkyl (4-trifluoromethylphenylamino)-(4-trifluoromethyl or 3-fluorophenyl) methylphosphonates

459

Synthesis and biological activities of novel isoxazoline-linked pseudodisaccharide derivatives Original Research Article

460

Synthesis and biological activities of novel nonpeptide angiotensin II receptor antagonists based on benzimidazole derivatives bearing a heterocyclic ring Original Research Article

461

Synthesis and biological activities of novel structural analogues of 2-arachidonoylglycerol, an endogenous cannabinoid receptor ligand

462

Synthesis and biological activities of novel β-Carbolines as PDE5 inhibitors

463

Synthesis and biological activities of nucleoside–estradiol conjugates

464

Synthesis and biological activities of octyl 2,3,4-tri-O-sulfo-α-l-fucopyranosyl-(1 → 3)-2,4-di-O-sulfo-α-l-fucopyranosyl-(1 → 3)-2,4-di-O-sulfo-α-l-fucopyranosyl-(1 → 3)-2,4-di-O-sulfo-β-l-fucopyranoside Original Research Article

465

Synthesis and biological activities of octyl 2,3-di-O-sulfo-α-l-fucopyranosyl-(1 → 3)-2-O-sulfo-α-l-fucopyranosyl-(1 → 4)-2,3-di-O-sulfo-α-l-fucopyranosyl-(1 → 3)-2-O-sulfo-α-l-fucopyranosyl-(1 → 4)-2,3-di-O-sulfo-β-l-fucopyranoside Original Research Arti

466

Synthesis and biological activities of phenyl piperazine- based peptidomimetic growth hormone secretagogues

467

Synthesis and biological activities of phenylahistin derivatives Original Research Article

468

Synthesis and biological activities of phthalocyanine–estradiol conjugates

469

Synthesis and biological activities of position one and three transposed analogs of the opioid peptide YKFA

470

Synthesis and biological activities of potential metabolites of the non-nucleoside reverse transcriptase inhibitor Efavirenz

471

Synthesis and biological activities of quinazoline derivatives with ortho-phenol-quaternary ammonium salt groups Original Research Article

472

Synthesis and biological activities of quinazoline derivatives with ortho-phenol-quaternary ammonium salt groups Original Research Article

473

Synthesis and biological activities of reveromycin A and spirofungin A derivatives

474

Synthesis and Biological Activities of Some Benzimidazoles Derivatives

475

Synthesis and Biological Activities of Some New Derivatives Based on 5-Styryl-2-amino-1,3,4-thiadiazole

476

Synthesis and biological activities of some new dibenzopyranones and dibenzopyrans: search for potential oestrogen receptor agonists and antagonists Original Research Article

477

Synthesis and biological activities of spiroheterocyclic growth hormone secretagogues

478

Synthesis and biological activities of the tris-oxazole macrolactone analogs of mycalolides

479

Synthesis and biological activities of three sulfated sialyl Lex ganglioside analogues for clarifying the real carbohydrate ligand structure of L-selectin Original Research Article

480

Synthesis and biological activities of topoisomerase I inhibitors, 6-N-amino analogues of NB-506

481

Synthesis and biological activities of truncated acridone: Structure-activity relationship studies of cytotoxic 5-hydroxy-4-quinolone

482

Synthesis and biological activities of ykfa analogues: effects of position 4 substitutions and altered ring size on In vitro opioid activity

483

Synthesis and biological activity evaluation of lignan lactones derived from (−)-cubebin

484

Synthesis and biological activity of (+)-hedychilactone A and its analogs from (+)-sclareolide

485

Synthesis and biological activity of [Tic5] didemnin B

486

Synthesis and biological activity of 1,2,3,4-tetrahydroquinoline and 3,4-(1H)-dihydroquinolin-2-one analogs of retinoic acid

487

Synthesis and biological activity of 1-alkylcarbonylmethyl analogues of YM022

488

Synthesis and biological activity of 1-methyl-tryptophan-tirapazamine hybrids as hypoxia-targeting indoleamine 2,3-dioxygenase inhibitors Original Research Article

489

Synthesis and Biological Activity of 1-Phenylsulfonyl-4-Phenylsulfonylaminopyrrolidine Derivatives as Thromboxane A2 Receptor Antagonists Original Research Article

490

Synthesis and biological activity of 1β-methyl-2-[5′-isoxazoloethenylpyrrolidin-3′-ylthio]carbapenems

491

Synthesis and biological activity of 2,5-diaryl-3-methylpyrimido[4,5-c]quinolin-1(2H)-one derivatives Original Research Article

492

Synthesis and biological activity of 22-iodo- and (E)-20(22)-dehydro analogues of 1α,25-dihydroxyvitamin D3 Original Research Article

493

Synthesis and biological activity of 22-oxa CD-ring modified analogues of 1α,25-dihydroxyvitamin D3: cis-perhydrindane CE-ring analogues

494

Synthesis and biological activity of 22-oxa CD-ring modified analogues of 1α,25-dihydroxyvitamin D3: spiro[5.5]undecane CF-ring analogues

495

Synthesis and biological activity of 2-alkylated deoxyadenosine bisphosphate derivatives as P2Y1 receptor antagonists Original Research Article

496

Synthesis and biological activity of 2-alkylbenzimidazoles bearing a N-phenylpyrrole moiety as novel angiotensin II AT1 receptor antagonists

497

Synthesis and biological activity of 2-anilino-4-(1H-pyrrol-3-yl) pyrimidine CDK inhibitors

498

Synthesis and biological activity of 2-Carbomethoxy-3-catechol-8-azabicyclo[3.2.1]octanes

499

Synthesis and biological activity of 2-methyl-20-epi analogues of 1α,25-dihydroxyvitamin D3

500

Synthesis and biological activity of 3,3-Diamino-sulfonylacrylonitriles as novel inhibitors of glucose induced insulin secretion from beta cells Original Research Article

501

Synthesis and biological activity of 3,4-dihydroquinazolines for selective T-type Ca2+ channel blockers

502

Synthesis and biological activity of 3-hydroxy(phosphono)methyl-bearing phosphatidylinositol ether lipid analogues

503

Synthesis and biological activity of 3-substituted 3-desoxynaltrindole derivatives

504

Synthesis and biological activity of 4′,8-dihydroxyisoflavon-7-yl d-hexopyranosides

505

Synthesis and biological activity of 4′-azido- and 4′-trifluoracetamido-3′-chloro-3′-deamino-4′-deoxydaunorubicin

506

Synthesis and biological activity of 4′-methoxy derivatives of abscisic acid

507

Synthesis and biological activity of 4-alkoxy chalcones: potential hydrophobic modulators of p-glycoprotein-mediated multidrug resistance Original Research Article

508

synthesis and biological activity of 4-methyl-3,5-dioxane derivatives as thromboxane a2 receptor antagonists Original Research Article

509

Synthesis and biological activity of 5-[(2,5-dihydroxybenzyl)amino]salicylic acid analogs as inhibitors of EGF receptor-associated protein tyrosine kinase

510

Synthesis and biological activity of 5-aryl-4-(4-(5-methyl-1H-imidazol-4-yl)piperidin-1-yl)pyrimidine analogs as potent, highly selective, and orally bioavailable NHE-1 inhibitors

511

Synthesis and biological activity of 5-aza-ellipticine derivatives

512

Synthesis and biological activity of 5-heteroaryl benzodiazepines: analogues of YM022

513

Synthesis and biological activity of 5-methylidene 1,2-dihydrochromeno[3,4-f]quinoline derivatives as progesterone receptor modulators

514

Synthesis and biological activity of 5-substituted-2-amino-1,3,4-oxadiazole derivatives

515

Synthesis and biological activity of 8β-substituted hydrocodone indole and hydromorphone indole derivatives

516

Synthesis and biological activity of a bivalent nucleotide inhibitor of ribonucleotide reductase

517

Synthesis and biological activity of a new anti-factor Xa pentasaccharide with a C-interglycosidic bond

518

Synthesis and Biological Activity of a New Pt(II) Complex Involving 4-bromo-2,6-bis-hydroxymethyl-phenol and Nicotinamide

519

Synthesis and Biological Activity of a New Schiff Base Ligand Pyridazine Based

520

Synthesis and biological activity of a novel class of cephalosporins with a oxadiazolyl hydroxypyridone moiety at C-7

521

Synthesis and biological activity of a novel class of pyridazine analogues as non-competitive reversible inhibitors of protein tyrosine phosphatase 1B (PTP1B) Original Research Article

522

Synthesis and biological activity of a novel series of indole-derived PPARγ agonists

523

Synthesis and biological activity of a novel squalene epoxidase inhibitor, FR194738

524

Synthesis and biological activity of a series of 4-aryl substituted benz[b]azepines: Antagonists at the strychnine-insensitive glycine site

525

Synthesis and biological activity of a stereoisomeric mixture of the mating hormone of Phytophthora

526

Synthesis and biological activity of amide derivatives of nimbolide

527

Synthesis and biological activity of analogues of batzelladine F

528

Synthesis and biological activity of analogues of ptilomycalin A

529

Synthesis and biological activity of A-nor-paclitaxel analogues Original Research Article

530

Synthesis and biological activity of anthelmintic thiadiazoles using an AF-2 receptor binding assay

531

Synthesis and biological activity of anticoccidial agents: 5,6-Diarylimidazo[2,1-b][1,3]thiazoles

532

Synthesis and biological activity of artificial analogs of mycalamide A

533

Synthesis and Biological Activity of C-6 and C-7 Modified Paclitaxels

534

Synthesis and Biological Activity of Certain Mannich Bases Derivatives from 1, 2, 4-Triazoles

535

Synthesis and biological activity of cinnamaldehydes as angiogenesis inhibitors

536

Synthesis and biological activity of conformationally constrained sialyl Lewis X analogues with reduced carbohydrate character

537

Synthesis and biological activity of conformationally restricted gypsy moth pheromone mimics Original Research Article

538

Synthesis and biological activity of conformationally restricted tricyclic analogs of the hormone melatonin

539

Synthesis and biological activity of conjugates between paclitaxel and the cell delivery vector penetratin

540

Synthesis and biological activity of copper(II) mixed ligand complexes with thiophene-2-aldehyde thiosemicarbazone as the primary ligand

541

Synthesis and biological activity of cyclic analogues of MPPG and MCPG as metabotropic glutamate receptor antagonists

542

Synthesis and biological activity of cyclotetrapeptide analogues of the natural HDAC inhibitor FR235222 Original Research Article

543

Synthesis and biological activity of derivatives of tetrahydroacridine as acetylcholinesterase inhibitors

544

Synthesis and biological activity of diaryl ether inhibitors of malarial enoyl acyl carrier protein reductase. Part 2: 2′-Substituted triclosan derivatives

545

Synthesis and biological activity of enantiomeric pairs of 5-[(E)-cycloalk-2-enylidenemethyl]thiolactomycin congeners

546

Synthesis and biological activity of enantiomeric pairs of 5-vinylthiolactomycin congeners

547

Synthesis and biological activity of enantiomers of a conformationally restricted muscarone analog

548

Synthesis and biological activity of ester and ether analogues of α-galactosylceramide (KRN7000) Original Research Article

549

Synthesis and biological activity of ferrocenyl derivatives of the non-steroidal antiandrogens flutamide and bicalutamide

550

Synthesis and biological activity of fluorinated 2-amino-4-aryl-3,4-dihydro[1,3,5]triazino[1,2-a]benzimidazoles

551

Synthesis and biological activity of fluorinated 7-aryl-2-pyridyl-6,7-dihydro[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-amines

552

Synthesis and biological activity of fluoroquinolone-pyrrolo[2,1-c][1,4]benzodiazepine conjugates Original Research Article

553

Synthesis and biological activity of fluoro-substituted pyrrolo[2,3-d]pyrimidines: The development of potential positron emission tomography imaging agents for the corticotropin-releasing hormone type 1 receptor

554

Synthesis and biological activity of glutamic acid derivatives

555

Synthesis and biological activity of high-affinity retinoic acid receptor antagonists Original Research Article

556

Synthesis and biological activity of hydroxylated analogs of RCAI-80

557

Synthesis and biological activity of hydroxylated analogues of KRN7000 (α-galactosylceramide) Original Research Article

558

Synthesis and biological activity of isopentenyl diphosphate analogues Original Research Article

559

Synthesis and biological activity of isoprenoid bisphosphonates Original Research Article

560

Synthesis and biological activity of J-104,118, a novel, potent inhibitor of squalene synthase

561

Synthesis and Biological activity of kappa opioid receptor agonists. Part 2: Preparation of 3-aryl-2-pyridone analogues generated by solution- and solid-phase parallel synthesis methods

562

Synthesis and biological activity of KCB-328 and its analogues: Novel class III antiarrhythmic agents with little reverse frequency dependence

563

Synthesis and biological activity of lactones en route to Altohyrtin A

564

Synthesis and biological activity of macrocyclic inhibitors of hepatitis C virus (HCV) NS3 protease

565

Synthesis and biological activity of macrocyclic taxane analogues

566

Synthesis and biological activity of medium molecular weight polymers of camptothecin

567

Synthesis and Biological Activity of Methanesulfonamide Pyrimidine- and N-Methanesulfonyl Pyrrole-Substituted 3,5-Dihydroxy-6-heptenoates, a Novel Series of HMG-CoA Reductase Inhibitors Original Research Article

568

Synthesis and biological activity of mustard derivatives of combretastatins

569

Synthesis and biological activity of N,N-dialkylaminoalkyl-substituted bisindolyl and diphenyl pyrazolone derivatives Original Research Article

570

Synthesis and biological activity of N4-phenylsubstituted-6-(2,4-dichloro phenylmethyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamines as vascular endothelial growth factor receptor-2 inhibitors and antiangiogenic and antitumor agents Original Research Article

571

Synthesis and biological activity of N-Acylated ornithine analogues of daptomycin

572

Synthesis and biological activity of naphthalene analogues of phenstatins: Naphthylphenstatins

573

Synthesis and biological activity of N-aroyl-tetrahydro-γ-carbolines Original Research Article

574

Synthesis and biological activity of N-aryl-2-aminothiazoles: potent pan inhibitors of cyclin-dependent kinases

575

Synthesis and biological activity of new 1,4-benzodioxan-arylpiperazine derivatives. Further validation of a pharmacophore model for α1-adrenoceptor antagonists Original Research Article

576

Synthesis and biological activity of new 5-O-sugar modified ketolide and 2-fluoro-ketolide antibiotics

577

Synthesis and biological activity of new anti-inflammatory compounds containing the 1,4-benzodioxine and/or pyrrole system Original Research Article

578

Synthesis and biological activity of new bradykinin pseudopeptide B1 receptor agonists containing alkylic spacers

579

Synthesis and biological activity of new melatonin dimeric derivatives Original Research Article

580

Synthesis and biological activity of new quinoxaline antibiotics of echinomycin analogues

581

Synthesis and Biological Activity of New Series of N-[3-(1H-1,2,3-Benzotriazol-1-yl)propyl]-2-(substituted Phenyl)-3-Chloro-4-Oxo-1-Azetidinecarboxamide

582

Synthesis and biological activity of N-methylated analogs of endomorphin-2 Original Research Article

583

Synthesis and biological activity of nociceptin/orphanin FQ analogues substituted in position 7 or 11 with Cα,α-dialkylated amino acids Original Research Article

584

Synthesis and biological activity of nociceptin/orphanin FQ(1–13)NH2 analogues modified in 9 and/or 13 position

585

Synthesis and biological activity of novel 1,2-disubstituted benzene derivatives as factor Xa inhibitors Original Research Article

586

Synthesis and biological activity of novel 1,4-diazepane derivatives as factor Xa inhibitor with potent anticoagulant and antithrombotic activity Original Research Article

587

Synthesis and biological activity of novel 1β-Methylcarbapenems with oxyiminopyrrolidinylamide moiety

588

Synthesis and biological activity of novel 2-(3-trifluoromethylphenoxy)-4-trifluoromethylthiazole-5-carboxamide derivatives

589

Synthesis and biological activity of novel 2-methyl-4-trifluoromethyl-thiazole-5-carboxamide derivatives

590

Synthesis and biological activity of novel 3-(4-methylthio benzene sulfonyl)-2,4-dimethyl/2,4-diphenyl/4-methyl-2-phenyl/2-ethoxy-4-methyl/ 2, 4-diethoxy–1,5-benzothiazepines

591

Synthesis and biological activity of novel 3′-trifluoromethyl taxoids

592

Synthesis and biological activity of novel 4,4-difluorobenzazepine derivatives as non-peptide antagonists of the arginine vasopressin V1A receptor Original Research Article

593

Synthesis and biological activity of novel 4-phenyl-1,8-naphthyridin-2(1H)-on-3-yl ureas: Potent acyl-CoA:cholesterol acyltransferase inhibitor with improved aqueous solubility

594

Synthesis and biological activity of novel antibacterial quinazolines

595

Synthesis and biological activity of novel cyanoacrylates containing ferrocenyl moiety

596

Synthesis and biological activity of novel macrocyclic antifungals: acylated conjugates of the ornithine moiety of the lipopeptidolactone FR901469

597

Synthesis and biological activity of novel macrocyclic antifungals: modification of the tyrosine moiety of the lipopeptidolactone FR901469

598

Synthesis and biological activity of novel N′-tert-butyl-N′-substituted benzoyl-N-(substituted phenyl)aminocarbonylhydrazines and their derivatives

599

Synthesis and Biological Activity of Novel Neuroprotective Diketopiperazines Original Research Article

600

Synthesis and biological activity of novel penem sulfoxides and sulfones

601

Synthesis and biological activity of novel peptide mimetics as melanocortin receptor agonists

602

Synthesis and biological activity of novel platinum(II) complexes of glutamate tethered to hydrophilic hematoporphyrin derivatives

603

Synthesis and biological activity of novel potent endothelin-converting enzyme-1 inhibitors

604

Synthesis and biological activity of novel pyrimidinone containing thiazolidinedione derivatives Original Research Article

605

Synthesis and biological activity of novel series of 4-methoxy, and 4,9-dimethoxy-5-substituted furo[2,3-g]-1,2,3-benzoxathiazine-7,7-dioxide derivatives

606

Synthesis and biological activity of novel sialyl-lewisX conjugates

607

Synthesis and biological activity of novel thiazolidin-4-ones with a carbohydrate moiety Original Research Article

608

Synthesis and biological activity of novel thiazolidinediones

609

Synthesis and biological activity of novel thyroid hormone analogues: 5′-aryl substituted GC-1 derivatives Original Research Article

610

Synthesis and biological activity of novel tricyclic β-lactams

611

Synthesis and biological activity of novel α-substituted β-phenylpropionic acids having pyridin-2-ylphenyl moiety as antihyperglycemic agents Original Research Article

612

Synthesis and biological activity of N-terminal lipidated and/or fluorescently labeled conjugates of astressin as corticotropin releasing factor antagonists Original Research Article

613

Synthesis and biological activity of olomoucine II

614

Synthesis and biological activity of oxo-7H-benzo[e]perimidine-4-carboxylic acid derivatives as potent, nonpeptide corticotropin releasing factor (CRF) receptor antagonists

615

Synthesis and biological activity of P2–P4 azapeptidomimetic P1-argininal and P1-ketoargininamide derivatives: a novel class of serine protease inhibitors

616

Synthesis and biological activity of Para-substituted 3′-phenyl docetaxel analogs

617

Synthesis and biological activity of peptidyl aldehyde urokinase inhibitors

618

Synthesis and biological activity of phenoxyphenyl oxamic acid derivatives related to -thyronine

619

Synthesis and biological activity of phosphatidylinositol-3,4,5-trisphosphorothioate

620

Synthesis and biological activity of piperazine and diazepane amides that are histamine H3 antagonists and serotonin reuptake inhibitors

621

Synthesis and biological activity of piperazine-Based dual MMP-13 and TNF-α converting enzyme inhibitors

622

Synthesis and biological activity of polygalloyl-dendrimers as stable tannic acid mimics

623

Synthesis and biological activity of potent heterocyclic thiol-based inhibitors of endothelin-converting enzyme-1

624

Synthesis and biological activity of previtamin D3 analogues with A-ring modifications Original Research Article

625

Synthesis and biological activity of quinolinone and dihydroquinolinone p38 MAP kinase inhibitors

626

Synthesis and biological activity of retinoic acid receptor-α specific amides

627

Synthesis and biological activity of Schiff and Mannich bases bearing 2,4-dichloro-5-fluorophenyl moiety Original Research Article

628

Synthesis and biological activity of selective azasugar-based TACE inhibitors

629

Synthesis and biological activity of selective pipecolic acid-based TNF-α converting enzyme (TACE) inhibitors

630

Synthesis and biological activity of semipeptoid farnesyltransferase inhibitors Original Research Article

631

Synthesis and biological activity of simplified denoviose-coumarins related to novobiocin as potent inhibitors of heat-shock protein 90 (hsp90)

632

Synthesis and biological activity of siRNA and Etoposide with magnetic nanoparticles on drug resistance model MCF-7 Cells: Molecular docking study with MRP1 enzyme

633

Synthesis and biological activity of some 3-acryloxymethyl cephalosporins

634

SYNTHESIS AND BIOLOGICAL ACTIVITY OF SOME BARBITURIC ACID DERIVATIVES VIA SCHIFF΄ S BASES

635

Synthesis and biological activity of some known and putative duloxetine metabolites

636

Synthesis and Biological Activity of Some New 5-Sulphanyl- 4-nitroimidazole Derivatives

637

Synthesis and biological activity of some new flavonyl-2,4-thiazolidinediones Original Research Article

638

Synthesis and Biological activity of Some PyrroloPyrimidine Compounds

639

Synthesis and Biological activity of Some PyrroloPyrimidine Compounds

640

Synthesis and biological activity of some rigid analogues of flavone-8-acetic acid Original Research Article

641

Synthesis and biological activity of some structural modifications of pancratistatin

642

Synthesis and biological activity of some sulphonamoylazopyrazoles

643

Synthesis and biological activity of S-oxo-[(methylthio)-methyl]cysteinols

644

Synthesis and biological activity of stable and potent antitumor agents, aniline nitrogen mustards linked to 9-anilinoacridines via a urea linkage Original Research Article

645

Synthesis and biological activity of substituted 3-fluoro/3-trifluoromethyl 10H-phenothiazines, its ribofuranosides and sulfones

646

Synthesis and biological activity of substituted bis-(4-hydroxyphenyl)methanes as N-type calcium channel blockers

647

Synthesis and biological activity of sulphostin analogues, novel dipeptidyl peptidase IV inhibitors Original Research Article

648

Synthesis and biological activity of the 1α,25-dihydroxyvitamin D3 diastereomer with unnatural configuration at the rings C/D side-chain moiety

649

Synthesis and biological activity of the first cyclic biphalin analogues

650

Synthesis and biological activity of the neuronal calcium channel blocker 2-amino-1-(2,5-dimethoxyphenyl)-5-trifluoromethyl benzimidazole (NS-649)

651

Synthesis and biological activity of the new 5-fluorocytosine derivatives, 5′-deoxy-N-alkyloxycarbonyl-5-fluorocytosine-5′-carboxylic acid

652

Synthesis and biological activity of the tea catechin metabolites, M4 and M6 and their methoxy-derivatives

653

Synthesis and biological activity of trans-2,3-dihydroraloxifene

654

Synthesis and biological activity of tricyclic aryloimidazo-, pyrimido-, and diazepinopurinediones Original Research Article

655

Synthesis and biological activity of vicinal diaryl-substituted 1H-imidazoles

656

Synthesis and Biological Activity of Water-Soluble Maleimide Derivatives of the Anticancer Drug Carboplatin Designed as Albumin-Binding Prodrugs

657

Synthesis and biological activity of α,β,γ,δ-unsaturated aldehydes from diatoms

658

Synthesis and biological activity of α-aminoboronic acids, amine-carboxyboranes and their derivatives

659

Synthesis and biological activity of β-glucuronyl carbamate-based prodrugs of paclitaxel as potential candidates for ADEPT Original Research Article

660

Synthesis and biological activity research of novel ferrocenyl-containing thiazole imine derivatives

661

Synthesis and Biological Activity Study of New Some Schiff Bases Derived From D-Erythroascorbic Acid

662

Synthesis and Biological Activity study of some New Isonicotinic Acid Hydrazide (isoniazid) Derivatives

663

Synthesis and biological affinity of new imidazo- and indol-arylpiperazine derivatives: Further validation of a pharmacophore model for α1-adrenoceptor antagonists

664

Synthesis and biological assays of E-ring analogs of camptothecin and homocamptothecin Original Research Article

665

Synthesis and Biological Assessment of 2-Hydroxyiminoethanones as Anti- Inflammatory and β-Amyloid Aggregation Inhibitors

666

Synthesis and biological characterisation of [3H]BBL454, a new CCK2 selective radiolabelled agonist displaying original pharmacological properties

667

Synthesis and biological characterization of [3H] (2-amino-4,5,6,7-tetrahydrobenzo[b]thiophen-3-yl)-(4-chlorophenyl)-methanone, the first radiolabelled adenosine A1 allosteric enhancer

668

Synthesis and biological characterization of AQPazide, a novel biotinylated photoaffinity probe for the study of the human platelet throm☐ane A2 receptor

669

Synthesis and biological characterization of novel hybrid 7-{[2-(4-phenyl-piperazin-1-yl)-ethyl]-propyl-amino}-5,6,7,8-tetrahydro-naphthalen-2-ol and their heterocyclic bioisosteric analogues for dopamine D2 and D3 receptors Original Research Article

670

Synthesis and biological characterization of stable and radioiodinated (±)-trans-2-hydroxy-3P{4-(3-iodophenyl)piperidyl}-1,2,3,4-tetrahydronaphthalene (3-IBVM)

671

Synthesis and biological data of 4-amino-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid ethyl esters, a new series of A1-adenosine receptor (A1AR) ligands

672

Synthesis and Biological Effectiveness of Some new Azo Compounds as Derivatives of Nitrogen Bases

673

Synthesis and biological effects of a new series of 2-amino-3-benzoylthiophenes as allosteric enhancers of A1-adenosine receptor

674

Synthesis and biological evaluation of - and -configuration 1,3-dioxolane 5-azacytosine and 6-azathymine nucleosides

675

Synthesis and biological evaluation of - and -configurations of 2′,3′-dideoxy-4′-c-methyl-3′-oxacytidine analogues

676

Synthesis and biological evaluation of (−)-dictyostatin and stereoisomers

677

Synthesis and biological evaluation of (−)-laulimalide analogues

678

Synthesis and biological evaluation of (±)-cryptotanshinone and its simplified analogues as potent CDC25 inhibitors

679

Synthesis and biological evaluation of (2S)- and (2R)-2-(3′-phosphonobicyclo[1.1.1]pentyl)glycines as novel group III selective metabotropic glutamate receptor ligands

680

Synthesis and biological evaluation of (3,4,5-trimethoxyphenyl)indol-3-ylmethane derivatives as potential antivascular agents Original Research Article

681

Synthesis and biological evaluation of (phenylpiperazinyl-propyl)arylsulfonamides as selective 5-HT2A receptor antagonists Original Research Article

682

Synthesis and biological evaluation of (R)-N-(diarylmethylthio/sulfinyl)ethyl/propyl-piperidine-3-carboxylic acid hydrochlorides as novel GABA uptake inhibitors

683

Synthesis and biological evaluation of [4-(2-phenylethenesulfonylmethyl)phenyl]-quinazolin-4-yl-amines as orally active anti-cancer agents

684

Synthesis and biological evaluation of 1-(2,4,5-trisubstituted phenyl)-3-(5-cyanopyrazin-2-yl)ureas as potent Chk1 kinase inhibitors

685

Synthesis and biological evaluation of 1-(4-[18f]fluorobenzyl)-4-[(5,6-dimethoxy-1-oxoindan2-yl)methyl]piperidine for in vivo studies of acetylcholinesterase

686

Synthesis and biological evaluation of 1-(benzenesulfonamido)-2-[5-(N-hydroxypyridin-2(1H)-one)]acetylene regioisomers: A novel class of 5-lipoxygenase inhibitors

687

Synthesis and biological evaluation of 1,1-Dichloro-2,3-diarylcyclopropanes as antitubulin and anti-breast cancer agents Original Research Article

688

Synthesis and biological evaluation of 1,1-difluoro-2-(tetrahydro-3-furanyl)ethylphosphonic acids possessing a N9-purinylmethyl functional group at the ring. A new class of inhibitors for purine nucleoside phosphorylases

689

Synthesis and biological evaluation of 1,2-disubstituted carbonucleosides of 2-amino-6-substituted purine and 8-azapurine

690

Synthesis and biological evaluation of 1,3,4-triaryl-3-pyrrolin-2-ones, a new class of selective cyclooxygenase-2 inhibitors

691

Synthesis and biological evaluation of 1,3-diphenylprop-2-en-1-ones possessing a methanesulfonamido or an azido pharmacophore as cyclooxygenase-1/-2 inhibitors Original Research Article

692

Synthesis and biological evaluation of 1,3-diphenylprop-2-yn-1-ones as dual inhibitors of cyclooxygenases and lipoxygenases

693

Synthesis and biological evaluation of 1,4-dihydropyridine calcium channel modulators having a diazen-1-ium-1,2-diolate nitric oxide donor moiety for the potential treatment of congestive heart failure Original Research Article

694

Synthesis and biological evaluation of 1,8-naphthyridin-4(1H)-on-3-carboxamide derivatives as new ligands of cannabinoid receptors Original Research Article

695

Synthesis and biological evaluation of 11C-labeled β-galactosyl triazoles as potential PET tracers for in vivo LacZ reporter gene imaging Original Research Article

696

Synthesis and biological evaluation of 12 allenic aromatic ethers

697

Synthesis and biological evaluation of 14-(aminoalkyl-aminomethyl)aromathecins as topoisomerase I inhibitors: Investigating the hypothesis of shared structure–activity relationships Original Research Article

698

Synthesis and biological evaluation of 14,15-dehydro-LTA4 analog

699

Synthesis and biological evaluation of 14-alkoxymorphinans. 14.1 14-ethoxy-5-methyl substituted indolomorphinans with δ opioid receptor selectivity

700

Synthesis and biological evaluation of 14-alkoxymorphinans.12.1 A phenethyl analogue of the μ-selective opioid receptor antagonist cyprodime

701

Synthesis and biological evaluation of 1-amino-1,1-bisphosphonates derived from fatty acids against Trypanosoma cruzi targeting farnesyl pyrophosphate synthase

702

Synthesis and biological evaluation of 1-azabicyclo-[3.2.1]octanes: new dopamine transporter inhibitors

703

Synthesis and biological evaluation of 1-benzyl-5-(3-biphenyl-2-yl-propyl)-1H-imidazole as novel farnesyltransferase inhibitor

704

Synthesis and biological evaluation of 1α,24-dihydroxy-25-nitrovitamin D3

705

Synthesis and biological evaluation of 1α-hydroxy-25(R and S)-25,26-Epoxy-23-yne vitamin D3 and of 1α,25(R and S),26-Trihydroxy-23-yne vitamin D3

706

Synthesis and biological evaluation of 2-(3′,4′,5′-trimethoxybenzoyl)-3-N,N-dimethylamino benzo[b]furan derivatives as inhibitors of tubulin polymerization Original Research Article

707

Synthesis and biological evaluation of 2-(4-fluorophenoxy)-2-phenyl-ethyl piperazines as serotonin-selective reuptake inhibitors with a potentially improved adverse reaction profile Original Research Article

708

Synthesis and biological evaluation of 2,2-disubstituted 2-aminoethanols: analogues of FTY720

709

Synthesis and biological evaluation of 2,3,4-triarylbenzopyran derivatives as SERM and therapeutic agent for breast cancer Original Research Article

710

Synthesis and biological evaluation of 2,3-diarylpyrazines and quinoxalines as selective COX-2 inhibitors Original Research Article

711

Synthesis and biological evaluation of 2,3-diarylthiophenes as selective Cox-2 and Cox-1 inhibitors

712

Synthesis and biological evaluation of 2,3-diarylthiophenes as selective cox-2 inhibitors. part II: Replacing the heterocycle

713

Synthesis and biological evaluation of 2,5-dihydropyrazolo[4,3-c]quinolin-3-ones, a novel series of PDE 4 inhibitors with low emetic potential and antiasthmatic properties

714

Synthesis and biological evaluation of 2,6-di-tert-butylphenol hydrazones as 5-lipoxygenase inhibitors Original Research Article

715

Synthesis and biological evaluation of 2,7-Dihydro-3H-dibenzo[de,h]cinnoline-3,7-dione derivatives, a novel group of anticancer agents active on a multidrug resistant cell line Original Research Article

716

Synthesis and biological evaluation of 2,8-disubstituted 9-benzyladenines: discovery of 8-mercaptoadenines as potent interferon-inducers Original Research Article

717

Synthesis and biological evaluation of 2′,5′-dimethoxychalcone derivatives as microtubule-targeted anticancer agents Original Research Article

718

Synthesis and biological evaluation of 2-alkylaminoethyl-1,1-bisphosphonic acids against Trypanosoma cruzi and Toxoplasma gondii targeting farnesyl diphosphate synthase Original Research Article

719

Synthesis and biological evaluation of 2-amino-2-deoxy- and 6-amino-6-deoxy-cyclomaltoheptaose polysulfates as synergists for angiogenesis inhibition Original Research Article

720

Synthesis and biological evaluation of 2-amino-3-(3′,4′,5′-trimethoxybenzoyl)-6-substituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine derivatives as antimitotic agents and inhibitors of tubulin polymerization

721

Synthesis and Biological Evaluation of 2-Aminothiazole Analogues of Nα-Protected Amino Acids

722

Synthesis and biological evaluation of 2-aminothiazoles and their amide derivatives on human adenosine receptors. Lack of effect of 2-aminothiazoles as allosteric enhancers Original Research Article

723

Synthesis and biological evaluation of 2-Hydroxy derivatives of digitoxigenin and 3-Epidigitoxigenin Original Research Article

724

Synthesis and Biological Evaluation of 2-Indolyloxazolines as a New Class of Tubulin Polymerization Inhibitors. Discovery of A-289099 as an Orally Active Antitumor Agent

725

Synthesis and biological evaluation of 2-methoxy- and 2-Methylthio-6-[(2′-alkylamino)ethyl]-4(3H)-pyrimidinones with anti-rubella virus activity Original Research Article

726

Synthesis and Biological Evaluation of 2-Phenyl Benzothiazole Derivatives as Cytotoxic Agents

727

Synthesis and biological evaluation of 2-thiopyrimidine derivatives Original Research Article

728

Synthesis and biological evaluation of 2-trifluoromethyl/sulfonamido-5,6-diaryl substituted imidazo[2,1-b]-1,3,4-thiadiazoles: A novel class of cyclooxygenase-2 inhibitors Original Research Article

729

Synthesis and biological evaluation of 2β,3α-(substituted phenyl)nortropanes as potential norepinephrine transporter imaging agents

730

Synthesis and biological evaluation of 3,4-diaryl-5-aminoisoxazole derivatives Original Research Article

731

Synthesis and biological evaluation of 3,4-diphenyl-1,2,5-oxadiazole-2-oxides and 3,4-diphenyl-1,2,5-oxadiazoles as potential hybrid COX-2 inhibitor/nitric oxide donor agents Original Research Article

732

Synthesis and biological evaluation of 3,5-diaminoindazoles as cyclin-dependent kinase inhibitors

733

Synthesis and biological evaluation of 3′,4′,5′-trimethoxychalcone analogues as inhibitors of nitric oxide production and tumor cell proliferation Original Research Article

734

Synthesis and biological evaluation of 3′-Carboranyl thymidine analogues

735

Synthesis and biological evaluation of 3-arylisoquinolines as antitumor agents

736

Synthesis and biological evaluation of 3-aryltyramines as fragments binding to BACE-1 and BACE-2

737

Synthesis and biological evaluation of 3-benzyl-1-methyl- and 1-methyl-3-phenyl-isothioureas as potential inhibitors of iNOS

738

Synthesis and biological evaluation of 3-ethylidene-1,3-dihydro-indol-2-ones as novel checkpoint 1 inhibitors

739

Synthesis and biological evaluation of 3-heteroaryloxy-4-phenyl-2(5H)-furanones as selective COX-2 inhibitors

740

Synthesis and biological evaluation of 3-substituted4-[2-(4"-isobutylphenyl)propionamido]-5-mercapto-l, 2,4-triazoles and their derivatives

741

Synthesis and biological evaluation of 4(5)-(6-methylpyridin-2-yl)imidazoles and -pyrazoles as transforming growth factor-β type 1 receptor kinase inhibitors Original Research Article

742

Synthesis and biological evaluation of 4-(hydroxyimino)arylmethyl diarylpyrimidine analogues as potential non-nucleoside reverse transcriptase inhibitors against HIV Original Research Article

743

Synthesis and biological evaluation of 4-[(3-Methyl-3H-imidazol-4-yl)-(2-phenylethynyl-benzyloxy)-methyl]-benzonitrile as novel farnesyltransferase inhibitor

744

Synthesis and biological evaluation of 4-[3-biphenyl-2-yl-1-hydroxy-1-(3-methyl-3H-imidazol-4-yl)-prop-2-ynyl]-1-yl-benzonitrile as novel farnesyltransferase inhibitor

745

Synthesis and biological evaluation of 4′-(6,7-disubstituted-2,4-dihydro-indeno[1,2-c]pyrazol-3-yl)-biphenyl-4-ol as potent Chk1 inhibitors

746

Synthesis and biological evaluation of 4-alkoxy substituted trinems. Part I

747

Synthesis and biological evaluation of 4-alkoxysubstituted trinems. Part II

748

Synthesis and biological evaluation of 4-amino derivatives of benzimidazoquinoxaline, benzimidazoquinoline, and benzopyrazoloquinazoline as potent IKK inhibitors

749

Synthesis and biological evaluation of 4-aryl-5-cyano-2H-1,2,3-triazoles as inhibitor of HER2 tyrosine kinase Original Research Article

750

Synthesis and biological evaluation of 4-Deacetoxy-1,7-dideoxy azetidine paclitaxel analogues

751

Synthesis and biological evaluation of 4-fluoroproline and 4-fluoropyrrolidine-2-acetic acid derivatives as new GABA uptake inhibitors Original Research Article

752

Synthesis and biological evaluation of 4-heterotribactams

753

Synthesis and Biological Evaluation of 4-hydroxychromenyl arylmethyl-6- hydroxy pyrimidine-2, 4-dione Derivatives

754

Synthesis and biological evaluation of 4-imidazolylflavans as nonsteroidal aromatase inhibitors

755

Synthesis and biological evaluation of 4-morpholino-2-phenylquinazolines and related derivatives as novel PI3 kinase p110α inhibitors Original Research Article

756

Synthesis and biological evaluation of 5-(pyridin-2-yl)thiazoles as transforming growth factor-β type1 receptor kinase inhibitors

757

Synthesis and biological evaluation of 5,6-diarylimidazo[2.1-b]thiazole as selective COX-2 inhibitors

758

Synthesis and biological evaluation of 5-[(aryl)(1H-imidazol-1-yl)methyl]-1H-indoles: Potent and selective aromatase inhibitors

759

Synthesis and biological evaluation of 5′-O-dicarboxylic fatty acyl monoester derivatives of anti-HIV nucleoside reverse transcriptase inhibitors

760

Synthesis and biological evaluation of 5-arylamino-1H-benzo[d]imidazole-4,7-diones as inhibitor of endothelial cell proliferation Original Research Article

761

Synthesis and biological evaluation of 5-arylamino-6-chloro-1H-indazole-4,7-diones as inhibitors of protein kinase B/Akt

762

Synthesis and biological evaluation of 5R- and 5S-methyl substituted d- and l-configuration 1,3-dioxolane nucleoside analogs Original Research Article

763

Synthesis and biological evaluation of 5-substituted 1,4-dihydroindeno[1,2-c]pyrazoles as multitargeted receptor tyrosine kinase inhibitors

764

Synthesis and biological evaluation of 5-substituted and 4,5-disubstituted-2-arylamino oxazole TRPV1 antagonists Original Research Article

765

Synthesis and biological evaluation of 6,7-disubstituted 4-aminopyrido[2,3-d]pyrimidines as adenosine kinase inhibitors

766

Synthesis and biological evaluation of 6′,7′-dihydroxybergamottin (6,7-DHB), a naturally occurring inhibitor of cytochrome P450 3A4

767

Synthesis and biological evaluation of 6-aryl-6H-pyrrolo[3,4-d]pyridazine derivatives as high-affinity ligands of the α2δ subunit of voltage-gated calcium channels

768

Synthesis and biological evaluation of 6-aryl-6H-pyrrolo[3,4-d]pyridazine derivatives: high-affinity ligands to the α2δ subunit of voltage gated calcium channels

769

Synthesis and biological evaluation of 6-oxa-nor-tropane glycomimetics as glycosidase inhibitors

770

Synthesis and biological evaluation of 7-azaindole derivatives, synthetic cytokinin analogues

771

Synthesis and biological evaluation of 7-azaindolocarbazoles

772

Synthesis and biological evaluation of 9-(5′,5′-difluoro-5′-phosphonopentyl)guanine derivatives for PNP-inhibitors Original Research Article

773

Synthesis and biological evaluation of 99mTc(CO)3-OH-PP-CS2 for brain receptor imaging

774

Synthesis and biological evaluation of 99mTc, Re-monoamine-monoamide conjugated to 2-(4-aminophenyl)benzothiazole as potential probes for β-amyloid plaques in the brain

775

Synthesis and biological evaluation of 9-deazaguanine derivatives connected by a linker to difluoromethylene phosphonic acid as multi-substrate analogue inhibitors of PNP

776

Synthesis and biological evaluation of 9-substituted tetracycline derivatives

777

Synthesis and biological evaluation of a 2-aryl polyhydroxylated pyrrolidine alkaloid-based library Original Research Article

778

Synthesis and biological evaluation of a bicyclo [7.4.1]enediyne

779

Synthesis and biological evaluation of a C5-biphenyl thiolactomycin library

780

Synthesis and biological evaluation of a conformationally free seco-analogue of the immunosuppressant FR901483 Original Research Article

781

Synthesis and biological evaluation of a des-dihydropyran laulimalide analog

782

SYNTHESIS AND BIOLOGICAL EVALUATION OF A FLUORINATED ANALOG OF THE β-ADRENERGIC BLOCKING AGENT, METOPROLOL

783

Synthesis and biological evaluation of a focused library of beauveriolides

784

Synthesis and Biological Evaluation of a New Benzofuran Analogue of 8-HETE

785

Synthesis and biological evaluation of a new class of bryostatin analogues: the role of the C20 substituent in protein kinase C binding

786

Synthesis and biological evaluation of a new class of bryostatin analogues: the role of the C20 substituent in protein kinase C binding

787

Synthesis and biological evaluation of a new class of bryostatin analogues: the role of the C20 substituent in protein kinase C binding

788

Synthesis and biological evaluation of a new class of vaccine adjuvants: aminoalkyl glucosaminide 4-phosphates (AGPs)

789

Synthesis and biological evaluation of a new series of berberine derivatives as dual inhibitors of acetylcholinesterase and butyrylcholinesterase Original Research Article

790

Synthesis and biological evaluation of a new series of dihydrofolate reductase inhibitors based on the 4-(2,6-diamino-5-pyrimidinyl)alkyl-L-glutamic acid structure

791

Synthesis and biological evaluation of a novel decadentate ligand DEPA

792

Synthesis and biological evaluation of a novel Glucosylated Derivative of Gadolinium Diethylenetriaminepentaacetic acid for Tumor Magnetic Resonance Imaging

793

Synthesis and biological evaluation of a novel phenyl substituted sydnone series as potential antitumor agents

794

SYNTHESIS an‎d BIOLOGICAL EVALUATION OF A NOVEL SERIES OF 2-(4-CHLORO-3-METHYLPHENOXY)ACETYL AMINO ACIDS an‎d PEPTIDES

795

Synthesis and biological evaluation of a novel series of pyrazole chalcones as anti-inflammatory, antioxidant and antimicrobial agents Original Research Article

796

Synthesis and biological evaluation of a novel structural type of serotonin 5-HT3 receptor antagonists

797

Synthesis and biological evaluation of a radiolabeled analog of methyl 2-acetamido-2,4-dideoxy-β-d-xylo-hexopyranoside directed towards influencing cellular glycosaminoglycan biosynthesis Original Research Article

798

Synthesis and biological evaluation of a series of 2′-fluorinated-2′,3′-dideoxy-2′,3′-didehydro-( )-nucleosides

799

Synthesis and biological evaluation of a series of A,B-ring modified 16,17-secoandrostane derivatives

800

Synthesis and biological evaluation of a series of flavone derivatives as potential radioligands for imaging the multidrug resistance-associated protein 1 (ABCC1/MRP1) Original Research Article

801

Synthesis and biological evaluation of a series of novel N- or O-fluoroalkyl derivatives of tropane: potential positron emission tomography (PET) imaging agents for the dopamine transporter

802

Synthesis and biological evaluation of a sialyl lewis X mimic with significantly improved E-selectin inhibition

803

Synthesis and biological evaluation of a small library of nojirimycin-derived bicyclic iminosugars Original Research Article

804

Synthesis and biological evaluation of a spongistatin AB-spiroketal analogue

805

Synthesis and biological evaluation of a technetium-99m(I)-tricarbonyl-labelled phenyltropane derivative

806

Synthesis and biological evaluation of a water soluble phosphate prodrug of 3-aminopyridine-2-carboxaldehyde thiosemicarbazone (3-AP)

807

Synthesis and biological evaluation of acyclic triaryl (Z)-olefins possessing a 3,5-di-tert-butyl-4-hydroxyphenyl pharmacophore: Dual inhibitors of cyclooxygenases and lipoxygenases Original Research Article

808

Synthesis and biological evaluation of aeroplysinin analogues: a new class of receptor tyrosine kinase inhibitors Original Research Article

809

Synthesis and biological evaluation of alkoxycoumarins as novel nematicidal constituents

810

Synthesis and biological evaluation of all A-ring stereoisomers of 5,6-trans-2-methyl-1,25-dihydroxyvitamin D3 and their 20-epimers: possible binding modes of potent A-ring analogues to vitamin D receptor Original Research Article

811

Synthesis and biological evaluation of allenic quinazolines using palladium-catalyzed hydride-transfer reaction

812

Synthesis and biological evaluation of amino-pyridines as androgen receptor antagonists for stimulating hair growth and reducing sebum production

813

Synthesis and biological evaluation of an 123I-labeled bicyclic nucleoside analogue (BCNA) as potential SPECT tracer for VZV-tk reporter gene imaging

814

Synthesis and biological evaluation of an alkenyldiarylmethane (ADAM) which acts as a novel non-nucleoside HIV-1 reverse transcriptase inhibitor

815

Synthesis and biological evaluation of an electronically activated isooxacephem Original Research Article

816

Synthesis and biological evaluation of an N10-Psec substituted pyrrolo[2,1-c][1,4]benzodiazepine prodrug

817

Synthesis and biological evaluation of an orally active ghrelin agonist that stimulates food consumption and adiposity in rats

818

Synthesis and biological evaluation of analogs of altohyrtin C (spongistatin 2)

819

Synthesis and biological evaluation of analogs of the marine toxin polycavernoside A

820

Synthesis and biological evaluation of analogues of bacterial lipid I

821

Synthesis and biological evaluation of analogues of the anti-tumor alkaloid naamidine A

822

Synthesis and biological evaluation of antitumor-active γ-butyrolactone substituted betulin derivatives Original Research Article

823

Synthesis and biological evaluation of antitumour-active betulin derivatives Original Research Article

824

Synthesis and biological evaluation of a-Ring biaryl-carbamate analogues of rhazinilam Original Research Article

825

Synthesis and biological evaluation of aristolactams

826

Synthesis and biological evaluation of aromatic enones related to curcumin Original Research Article

827

Synthesis and biological evaluation of aroylguanidines related to amiloride as inhibitors of the human platelet Na+/H+ exchanger Original Research Article

828

Synthesis and biological evaluation of aryl azide derivatives of combretastatin a-4 as molecular probes for tubulin Original Research Article

829

Synthesis and biological evaluation of asymmetric gramicidin S analogues containing modified d-phenylalanine residues Original Research Article

830

Synthesis and biological evaluation of aziridine-containing analogs of phytosphingosine

831

Synthesis and biological evaluation of bengacarboline derivatives

832

Synthesis and biological evaluation of benzamides and benzamidines as selective inhibitors of VEGFR tyrosine kinases

833

Synthesis and biological evaluation of benzamides and benzamidines: structural requirement of a pyrimidine ring for inhibition of EGFR tyrosine kinase

834

Synthesis and biological evaluation of benzazepine oxazolidinone antibacterials

835

Synthesis and biological evaluation of benzimidazole derivatives as potent AMP-activated protein kinase activators Original Research Article

836

Synthesis and biological evaluation of benzimidazole-4,7-diones that inhibit vascular smooth muscle cell proliferation

837

Synthesis and biological evaluation of benzo[b]naphthyridones, a series of new topical antibacterial agents

838

Synthesis and biological evaluation of benzoic acid derivatives as potent, orally active VLA-4 antagonists Original Research Article

839

Synthesis and biological evaluation of benzopyran analogues bearing class III antiarrhythmic pharmacophores Original Research Article

840

Synthesis and biological evaluation of benzothiazole derivatives as potent antitumor agents

841

Synthesis and biological evaluation of bicyclic and tricyclic substituted nortropane derivatives: discovery of a novel selective α1D-adrenergic receptor ligand Original Research Article

842

Synthesis and biological evaluation of bidentate 3-hydroxypyridin-4-ones iron chelating agents

843

Synthesis and biological evaluation of biphenylsulfonamide carboxylate aggrecanase-1 inhibitors

844

Synthesis and biological evaluation of bis and monocarbonate prodrugs of 10-hydroxycamptothecins Original Research Article

845

Synthesis and biological evaluation of both enantiomers of L-761,000 as inhibitors of cyclooxygenase 1 and 2

846

Synthesis and biological evaluation of branched and conformationally restricted analogs of the anticancer compounds 3′-C-ethynyluridine (EUrd) and 3′-C-ethynylcytidine (ECyd) Original Research Article

847

Synthesis and biological evaluation of B-ring analogues of (−)-rhazinilam Original Research Article

848

Synthesis and biological evaluation of B-ring modified colchicine and isocolchicine analogs

849

Synthesis and biological evaluation of bryostatin analogues: the role of the A-ring

850

Synthesis and biological evaluation of C-12′ substituted vinflunine derivatives

851

Synthesis and biological evaluation of carboacyclic nucleosides with (Z) and (E)-9-[4,4-bis(hydroxymethyl)]-2-butenyl side chain Original Research Article

852

Synthesis and biological evaluation of carbohydrate appended hydrazinocyclopentenes with potent glycation and α-glucosidase inhibition activities

853

Synthesis and biological evaluation of cepharadiones A and B and related dioxoaporphines Original Research Article

854

SYNTHESIS AND BIOLOGICAL EVALUATION OF CERTAIN 2H-PYRAN-2- ONES AND SOME DERIVED 1H-PYRIDIN-2-ONE ANALOGS AS ANTIMICROBIAL AGENTSa

855

Synthesis and Biological Evaluation of Certain New Substituted Pyrido[2,3-d]pyrimidin-4(1H)-one and Pyrido[2,3-d]triazolo[3,4-b]pyrimidine Analogs

856

Synthesis and biological evaluation of chalcones and their derived pyrazoles as potential cytotoxic agents

857

Synthesis and biological evaluation of chalcones as inhibitors of the voltage-gated potassium channel Kv1.3

858

Synthesis and biological evaluation of chromone carboxamides as calpain inhibitors

859

Synthesis and biological evaluation of cinnamyl compounds as potent antitumor agents

860

Synthesis and biological evaluation of clitocine analogues as adenosine kinase inhibitors

861

Synthesis and biological evaluation of conformationally constrained analogs of the antitumor agents XK469 and SH80. Part 5 Original Research Article

862

Synthesis and biological evaluation of conformationally constrained analogues of the antitubercular agent ethambutol Original Research Article

863

Synthesis and biological evaluation of conformationally constrained bicyclic and tricyclic balanol analogues as inhibitors of protein kinase C

864

Synthesis and biological evaluation of conformationally restricted gabapentin analogues

865

Synthesis and biological evaluation of copper (II) complexes of sterically hindered o-aminophenol derivatives as antimicrobial agents

866

Synthesis and biological evaluation of coumarincarboxylic acids as inhibitors of gyrase B. L-rhamnose as an effective substitute for L-noviose

867

Synthesis and biological evaluation of cremastrine and an unnatural analogue

868

Synthesis and biological evaluation of cryptophycin analogs with substitution at C-6 (fragment C region)

869

Synthesis and biological evaluation of CX-659S and its related compounds for their inhibitory effects on the delayed-type hypersensitivity reaction Original Research Article

870

Synthesis and biological evaluation of cyclic and branched peptide analogues as ligands for cholecystokinin type 1 receptor Original Research Article

871

Synthesis and biological evaluation of cyclopenta[c]thiophene related compounds as new antitumor agents Original Research Article

872

Synthesis and Biological Evaluation of Cyclophostin: A 5′,6″-Tethered Analog of Adenophostin A

873

Synthesis and Biological Evaluation of Cyclopropyl Analogs of the Antiestrogen MER 25

874

Synthesis and biological evaluation of cytostatin analogues

875

Synthesis and biological evaluation of cytotoxic activity of novel anthracene l-rhamnopyranosides Original Research Article

876

Synthesis and biological evaluation of deoxy salacinols, the role of polar substituents in the side chain on the α-glucosidase inhibitory activity Original Research Article

877

Synthesis and biological evaluation of deoxypreussomerin A and palmarumycin CP1 and related naphthoquinone spiroketals

878

Synthesis and biological evaluation of diamine-based histamine H3 antagonists with serotonin reuptake inhibitor activity

879

Synthesis and biological evaluation of didemnin photoaffinity analogues

880

Synthesis and biological evaluation of dihydrofuran-fused perhydrophenanthrenes as a new anti-influenza agent having novel structural characteristic Original Research Article

881

Synthesis and biological evaluation of dimeric cinnamaldehydes as potent antitumor agents Original Research Article

882

Synthesis and biological evaluation of disubstituted N6-cyclopentyladenine analogues: the search for a neutral antagonist with high affinity for the adenosine A1 receptor Original Research Article

883

Synthesis and biological evaluation of DNA targeting flexible side-chain substituted β-carboline derivatives

884

Synthesis and biological evaluation of enantiopure thionitrites: The solid-phase synthesis and nitrosation of -glutathione as a molecular probe

885

Synthesis and biological evaluation of epothilone A dimeric compounds Original Research Article

886

Synthesis and biological evaluation of ether bridged bicyclic iminosugar derivatives Original Research Article

887

Synthesis and biological evaluation of fenobam analogs as mGlu5 receptor antagonists

888

Synthesis and Biological Evaluation of Five- and Six-Membered Heterocycles as an Anti-Diabetic Agent: An Overview

889

Synthesis and biological evaluation of five-Membered heterocycles fused to cyclopenta[c]thiophene as new antitumor agents Original Research Article

890

Synthesis and biological evaluation of flavan-3-ol derivatives as positive modulators of GABAA receptors Original Research Article

891

Synthesis and biological evaluation of flavonoids and related compounds as gastroprotective agents

892

Synthesis and Biological Evaluation of Flavonoids as Antiacetylcholinesterase Agent

893

Synthesis and biological evaluation of flavonoids as vasorelaxant agents

894

Synthesis and biological evaluation of fluorescently labeled epothilone analogs for tubulin binding studies

895

Synthesis and biological evaluation of fluorinated acyclothionucleosides

896

Synthesis and biological evaluation of four stereoisomers of PDMP-analogue, N-(2-decylamino-3-hydroxy-3-phenylprop-1-yl)-β-valienamine, and related compounds

897

Synthesis and biological evaluation of GABA derivatives able to cross the blood–Brain barrier in rats

898

Synthesis and biological evaluation of galactofuranosyl alkyl thioglycosides as inhibitors of mycobacteria Original Research Article

899

Synthesis and biological evaluation of gambierol analogues

900

Synthesis and biological evaluation of gemcitabine–lipid conjugate (NEO6002)

901

Synthesis and biological evaluation of gem-diamine 1-N-iminosugars related to l-iduronic acid as inhibitors of heparan sulfate 2-O-sulfotransferase

902

Synthesis and biological evaluation of glycal-derived novel tetrahydrofuran 1,2,3-triazoles by ‘click’ chemistry Original Research Article

903

Synthesis and biological evaluation of glycosylated psoralen derivatives

904

Synthesis and biological evaluation of guanylhydrazone coactivator binding inhibitors for the estrogen receptor Original Research Article

905

Synthesis and biological evaluation of helicid analogues as mushroom tyrosinase inhibitors

906

Synthesis and biological evaluation of heterocycle containing adamantane 11β-HSD1 inhibitors

907

Synthesis and biological evaluation of highly potent analogues of epothilones B and D

908

Synthesis and biological evaluation of histone deacetylase inhibitors that are based on FR235222: A cyclic tetrapeptide scaffold

909

Synthesis and biological evaluation of homopiperazine derivatives with β-aminoacyl group as dipeptidyl peptidase IV inhibitors

910

Synthesis and biological evaluation of homoserine lactone derived ureas as antagonists of bacterial quorum sensing Original Research Article

911

Synthesis and biological evaluation of hybrid molecules containing the pyrroloquinoline nucleus and DNA-minor groove binders

912

Synthesis and Biological Evaluation of Hydrazones fromNontraditional oils

913

Synthesis and biological evaluation of hydrophilic embelin derivatives

914

Synthesis and biological evaluation of hydroxamate-Based inhibitors of glutamate carboxypeptidase II

915

Synthesis and biological evaluation of imidazo[1,2-a]pyridine derivatives as novel PI3 kinase p110α inhibitors Original Research Article

916

Synthesis and biological evaluation of imidazol-2-one and 2-cyanoiminoimidazole derivatives: novel series of PDE4 inhibitors

917

Synthesis and biological evaluation of imidazol-2-one derivatives as potential antitumor agents Original Research Article

918

Synthesis and biological evaluation of imidazole thioacetanilides as novel non-nucleoside HIV-1 reverse transcriptase inhibitors Original Research Article

919

Synthesis and biological evaluation of imidazole-based small molecule antagonists of the melanocortin 4 receptor (MC4-R)

920

Synthesis and biological evaluation of immunosuppressive agent DZ2002 and its stereoisomers Original Research Article

921

Synthesis and biological evaluation of indazolo[4,3-bc][1,5]naphthyridines (10-aza-pyrazolo[3,4,5-kl]acridines): a new class of antitumor agents Original Research Article

922

Synthesis and biological evaluation of indolyl bisphosphonates as anti-bone resorptive and anti-leishmanial agents Original Research Article

923

Synthesis and biological evaluation of isoflavone analogues from Dalbergia oliveri

924

Synthesis and biological evaluation of isoflavone fatty acid esters with potential weight loss and hypolipidemic activities Original Research Article

925

Synthesis and biological evaluation of l-cysteine derivatives as mitotic kinesin Eg5 inhibitors

926

Synthesis and biological evaluation of linear phenylethynylbenzenesulfonamide regioisomers as cyclooxygenase-1/-2 (COX-1/-2) inhibitors Original Research Article

927

Synthesis and biological evaluation of lipophilic Ca1a2L analogues as potential bisubstrate inhibitors of protein:geranylgeranyl transferase-1 Original Research Article

928

Synthesis and biological evaluation of lisofylline (LSF) analogs as a potential treatment for Type 1 diabetes

929

Synthesis and biological evaluation of l-α-Phosphatidyl-d-3-deoxy-3-heteromethyl-myo-inositols as phosphoinositide 3-kinase inhibitors Original Research Article

930

Synthesis and Biological Evaluation of MAO-A Selective 1,4-Disubstituted-1,2,3,6-tetrahydropyridinyl Substrates Original Research Article

931

Synthesis and biological evaluation of menthol-based derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1)

932

Synthesis and biological evaluation of methoxylated analogs of the newer generation taxoids IDN5109 and IDN5390

933

Synthesis and biological evaluation of methoxyphenyl porphyrin derivatives as potential photodynamic agents Original Research Article

934

Synthesis and Biological Evaluation of Metronidazole Derivatives as Anti-Giardia Agents

935

Synthesis and biological evaluation of mixed ammine/amine platinum(II) complexes with dicarboxylate containing organic nitrate as ligand

936

Synthesis and biological evaluation of N-(1-aziridino)-6-fluoro-quinolone-3-carboxylic acids

937

Synthesis and Biological Evaluation of N-(5-(pyridin-2-yl)-1,3,4-thiadiazol- 2-yl)benzamide Derivatives as Lipoxygenase Inhibitor with Potential Anticancer Activity

938

Synthesis and biological evaluation of N-(7-indazolyl)benzenesulfonamide derivatives as potent cell cycle inhibitors Original Research Article

939

Synthesis and biological evaluation of N-(7-indolyl)-3-pyridinesulfonamide derivatives as potent antitumor agents

940

Synthesis and biological evaluation of N-(aryl)-2-thiophen-2-ylacetamides series as a new class of antitubercular agents

941

Synthesis and biological evaluation of N-{4-[5-(2,4-diamino-6-oxo-1,6-dihydropyrimidin-5-yl)-2-(2,2,2-trifluoroacetyl)pentyl]benzoyl}-l-glutamic acid as a potential inhibitor of GAR Tfase and the de novo purine biosynthetic pathway Original Research Artic

942

Synthesis and biological evaluation of N-acetyl-β-aryl-1,2-didehydroethylamines as new HIV-1 RT inhibitors in vitro

943

Synthesis and Biological Evaluation of New 1, 4-Dihydropyridines as Antihypertensives Agents in Rats

944

Synthesis and Biological Evaluation of New 1,4-Thiazine Containing Heterocyclic Compounds

945

Synthesis and biological evaluation of new 1,5-diazaanthraquinones with cytotoxic activity Original Research Article

946

Synthesis and biological evaluation of new 3,5-di(trifluoromethyl)-1,2,4-triazolesulfonylurea and thiourea derivatives as antidiabetic and antimicrobial agents

947

Synthesis and biological evaluation of new 3-substituted indole derivatives as potential anti-inflammatory and analgesic agents Original Research Article

948

Synthesis and biological evaluation of new 3-trifluoromethylpyrazolesulfonyl-urea and thiourea derivatives as antidiabetic and antimicrobial agents

949

Synthesis and biological evaluation of new 4-arylpiperidines and 4-aryl-4-piperidinols: dual Na+ and Ca2+ channel blockers with reduced affinity for dopamine D2 receptors Original Research Article

950

Synthesis and biological evaluation of new 4-carboxyl quinoline derivatives as cyclooxygenase-2 inhibitors Original Research Article

951

Synthesis and biological evaluation of new 4β-anilino- and 4β-imido-substituted podophyllotoxin congeners Original Research Article

952

Synthesis and biological evaluation of new 6-s-cis locked 1,2,25-trihydroxyprevitamin D3 analogues Original Research Article

953

Synthesis and biological evaluation of new antimalarial isonitriles related to marine diterpenoids

954

Synthesis and biological evaluation of new arylthiophene analogs of DuP 753

955

Synthesis and biological evaluation of new barbituric and thiobarbituric acid fluoro analogs of benzenesulfonamides as antidiabetic and antibacterial agents

956

Synthesis and biological evaluation of new biphalin analogues with non-hydrazine linkers

957

Synthesis and biological evaluation of new BSH-conjugated chlorin derivatives as agents for both photodynamic therapy and boron neutron capture therapy of cancer

958

Synthesis and biological evaluation of new conformationally biased integrin ligands based on a tetrahydroazoninone scaffold

959

Synthesis and biological evaluation of new derivatives of emodin Original Research Article

960

Synthesis and biological evaluation of new diisocyanide- and triisocyanide-99mTc complexes

961

Synthesis and biological evaluation of new dipyrrolo[3,4-a:3,4-c]carbazole-1,3,4,6-tetraones, substituted with various saturated and unsaturated side chains via palladium catalyzed cross-coupling reactions Original Research Article

962

Synthesis and biological evaluation of new disubstituted analogues of 6-methoxy-3-(3′,4′,5′-trimethoxybenzoyl)-1H-indole (BPR0L075), as potential antivascular agents Original Research Article

963

Synthesis and biological evaluation of new mannose 6-phosphate analogues Original Research Article

964

Synthesis and biological evaluation of new N-(2-hydroxy-4(or 5)-nitro/aminophenyl)benzamides and phenylacetamides as antimicrobial agents Original Research Article

965

Synthesis and Biological Evaluation of New Nitroimidazole Derivatives as Anti-Helicobacter pylori Agents Against Metronidazole-Resistant Strains

966

Synthesis and biological evaluation of new non-imidazole H3-receptor antagonists of the 2-aminobenzimidazole series Original Research Article

967

Synthesis and biological evaluation of new oxime-ether derivatives of steroid as anti-bacterial agents

968

Synthesis and biological evaluation of new pyrazole- and tetrazole-related C-nucleosides with modified sugar moieties

969

Synthesis and biological evaluation of new pyridines containing imidazole moiety as antimicrobial and anticancer agents

970

Synthesis and biological evaluation of new spin-labeled derivatives of podophyllotoxin Original Research Article

971

Synthesis and biological evaluation of new symmetrical derivatives as cytotoxic agents and apoptosis inducers Original Research Article

972

Synthesis and biological evaluation of new taxoids derived from 2-deacetoxytaxinine J

973

Synthesis and biological evaluation of new tetrahydronaphthalene derivatives as thromboxane receptor antagonists

974

Synthesis and biological evaluation of new tetrahydro-β-carbolines as inhibitors of the mitotic kinesin Eg5 Original Research Article

975

Synthesis and biological evaluation of new UDP-GalNAc analogues for the study of polypeptide-α-GalNAc-transferases

976

Synthesis and biological evaluation of N-heterocyclic carbene–silver(I) acetate complexes derived from 4,5-ditolyl-imidazole

977

Synthesis and biological evaluation of nitric oxide-releasing derivatives of oleanolic acid as inhibitors of HepG2 cell apoptosis

978

Synthesis and biological evaluation of N-mercaptoacylproline and N-mercaptoacylthiazolidine-4-carboxylic acid derivatives as leukotriene A4 hydrolase inhibitors

979

Synthesis and biological evaluation of N-methyl-laudanosine iodide analogues as potential SK channel blockers Original Research Article

980

Synthesis and Biological Evaluation of Nonionic Prenyl, Geranyl, and Farnesyl Diphosphate Surrogates

981

Synthesis and biological evaluation of nonpeptide integrin antagonists containing spirocyclic scaffolds

982

Synthesis and biological evaluation of nonpeptide mimetics of ω-conotoxin GVIA Original Research Article

983

Synthesis and biological evaluation of non-peptide αvβ3/α5β1 integrin dual antagonists containing 5,6-dihydropyridin-2-one scaffolds Original Research Article

984

Synthesis and biological evaluation of non-polyene analogs of amphotericin B

985

Synthesis and biological evaluation of norcantharidin analogues: Towards PP1 selectivity Original Research Article

986

Synthesis and Biological Evaluation of Novel -2′-Azido-2′,3′-dideoxyarabinofuranosyl-4′-thiopyrimidines and purines

987

Synthesis and biological evaluation of novel (4 or 5-aryl)pyrazolyl-indoles as inhibitors of interleukin-2 inducible T-cell kinase (ITK) Original Research Article

988

Synthesis and biological evaluation of novel (l)-α-amino acid methyl ester, heteroalkyl, and aryl substituted 1,4-naphthoquinone derivatives as antifungal and antibacterial agents

989

Synthesis and biological evaluation of novel 1,3,5-triazine derivatives as antimicrobial agents

990

Synthesis and biological evaluation of novel 1,4-naphthoquinone derivatives as antibacterial and antiviral agents

991

Synthesis and biological evaluation of novel 1,5-benzothiazepin-4(5H)-ones as potent antiangiogenic and antioxidant agents

992

Synthesis and biological evaluation of novel 1-O- and 14-O-derivatives of oridonin as potential anticancer drug candidates

993

Synthesis and biological evaluation of novel 1β-methylcarbapenems having a new moiety at C-2

994

Synthesis and biological evaluation of novel 1β-methylcarbapenems with isothiazoloethenyl side chains

995

Synthesis and biological evaluation of novel 2-(1H-imidazol-4-yl)cyclopropane carboxylic acids: key intermediates for H3 histamine receptor ligands

996

Synthesis and biological evaluation of novel 2-(substituted phenylaminocarbonylmethylthio)-6-(2,6-dichlorobenzyl)-pyrimidin-4(3H)-ones as potent HIV-1 NNRTIs Original Research Article

997

Synthesis and biological evaluation of novel 2′-deoxy-4′-thio-imidazole nucleosides Original Research Article

998

Synthesis and biological evaluation of novel 2-pyridinyl-[1,2,3]triazoles as inhibitors of transforming growth factor β1 type 1 receptor

999

Synthesis and biological evaluation of novel 2-vinyl carbapenems. Remarkable DHP-1 stability of 1′-substituted analogs

1000

Synthesis and biological evaluation of novel 3′-difluorovinyl taxoids

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